TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 220nMAssay Description:Competitive inhibition of Mycobacterium tuberculosis H37Rv PTP-B expressed in Escherichia coli DE3 using p-nitrophenyl phosphate as substrate preincu...More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase YopH(Yersinia enterocolitica)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 4.40E+3nMAssay Description:Competitive inhibition of Yersinia enterocolitica recombinant YopH using pNPP as substrate after 10 mins by Line-weaver Burk plot analysisMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase YopH(Yersinia enterocolitica)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 4.40E+3nMAssay Description:Competitive inhibition of Yersinia enterocolitica recombinant YopH using pNPP as substrate after 10 mins by Line-weaver Burk plot analysisMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase YopH(Yersinia enterocolitica)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 4.50E+3nMAssay Description:Competitive inhibition of Yersinia enterocolitica recombinant YopH using pNPP as substrate after 10 mins by Line-weaver Burk plot analysisMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 4.90E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PTPA-mediated pNPP hydrolysisMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 5.40E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PTPA-mediated pNPP hydrolysisMore data for this Ligand-Target Pair
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 8.00E+3nMAssay Description:Competitive inhibition of Mycobacterium tuberculosis PTP-B using p-nitrophenyl phosphate as substrate measured for 10 mins by Lineweaver-Burk plot an...More data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 9.10E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PTPA-mediated pNPP hydrolysisMore data for this Ligand-Target Pair
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 1.00E+4nMAssay Description:Competitive inhibition of Mycobacterium tuberculosis PTP-B using p-nitrophenyl phosphate as substrate measured for 10 mins by Lineweaver-Burk plot an...More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase YopH(Yersinia enterocolitica)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 1.11E+4nMAssay Description:Competitive inhibition of Yersinia enterocolitica recombinant YopH using pNPP as substrate after 10 mins by Line-weaver Burk plot analysisMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 1.20E+4nMAssay Description:Competitive inhibition of Mycobacterium tuberculosis PTP-A using p-nitrophenyl phosphate as substrate measured for 10 mins by Lineweaver-Burk plot an...More data for this Ligand-Target Pair
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 1.30E+4nMAssay Description:Competitive inhibition of Mycobacterium tuberculosis PTP-B using p-nitrophenyl phosphate as substrate measured for 10 mins by Lineweaver-Burk plot an...More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase YopH(Yersinia enterocolitica)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 1.41E+4nMAssay Description:Competitive inhibition of Yersinia enterocolitica recombinant YopH using pNPP as substrate after 10 mins by Line-weaver Burk plot analysisMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 1.79E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PTPA-mediated pNPP hydrolysisMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 2.13E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PTPA-mediated pNPP hydrolysisMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 2.30E+4nMAssay Description:Competitive inhibition of Mycobacterium tuberculosis PTP-A using p-nitrophenyl phosphate as substrate measured for 10 mins by Lineweaver-Burk plot an...More data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 2.90E+4nMAssay Description:Competitive inhibition of Mycobacterium tuberculosis PTP-A using p-nitrophenyl phosphate as substrate measured for 10 mins by Lineweaver-Burk plot an...More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase YopH(Yersinia enterocolitica)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataKi: 3.60E+4nMAssay Description:Noncompetitive inhibition of Yersinia enterocolitica recombinant YopH using pNPP as substrate after 10 mins by Line-weaver Burk plot analysisMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
School Of Health Sciences/Graduate Program In Pharmaceutical Sciences
Curated by ChEMBL
School Of Health Sciences/Graduate Program In Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
School Of Health Sciences/Graduate Program In Pharmaceutical Sciences
Curated by ChEMBL
School Of Health Sciences/Graduate Program In Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 52nMAssay Description:Inhibition of human acetylcholinesterase using acetylthiocholine iodide as substrate incubated for 15 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
School Of Health Sciences/Graduate Program In Pharmaceutical Sciences
Curated by ChEMBL
School Of Health Sciences/Graduate Program In Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 68nMAssay Description:Inhibition of human acetylcholinesterase using acetylthiocholine iodide as substrate incubated for 15 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
School Of Health Sciences/Graduate Program In Pharmaceutical Sciences
Curated by ChEMBL
School Of Health Sciences/Graduate Program In Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 87nMAssay Description:Inhibition of human acetylcholinesterase using acetylthiocholine iodide as substrate incubated for 15 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
School Of Health Sciences/Graduate Program In Pharmaceutical Sciences
Curated by ChEMBL
School Of Health Sciences/Graduate Program In Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 178nMAssay Description:Inhibition of human acetylcholinesterase using acetylthiocholine iodide as substrate incubated for 15 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
School Of Health Sciences/Graduate Program In Pharmaceutical Sciences
Curated by ChEMBL
School Of Health Sciences/Graduate Program In Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of human acetylcholinesterase using acetylthiocholine iodide as substrate incubated for 15 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Bmssi Umr 5086 Cnrs/Universit£
Curated by ChEMBL
Bmssi Umr 5086 Cnrs/Universit£
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of human ABCG2 ATPase activity transfected in Sf9 insect cells using quercetin as substrate after 30 mins by colorimetry relative to contr...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Bmssi Umr 5086 Cnrs/Universit£
Curated by ChEMBL
Bmssi Umr 5086 Cnrs/Universit£
Curated by ChEMBL
Affinity DataIC50: 270nMAssay Description:Inhibition of human ABCG2 ATPase activity transfected in Sf9 insect cells using quercetin as substrate after 30 mins by colorimetry relative to contr...More data for this Ligand-Target Pair
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataIC50: 440nMAssay Description:Inhibition of N-terminal histidine-tagged Mycobacterium tuberculosis PTPB expressed in Escherichia coli BL21 (DE3) after 45 mins by fluorescence assa...More data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Inhibition of HIV1 integrase strand transfer activityMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
School Of Health Sciences/Graduate Program In Pharmaceutical Sciences
Curated by ChEMBL
School Of Health Sciences/Graduate Program In Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 640nMAssay Description:Inhibition of human acetylcholinesterase using acetylthiocholine iodide as substrate incubated for 15 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
School Of Health Sciences/Graduate Program In Pharmaceutical Sciences
Curated by ChEMBL
School Of Health Sciences/Graduate Program In Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 799nMAssay Description:Inhibition of human acetylcholinesterase using acetylthiocholine iodide as substrate incubated for 15 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
School Of Health Sciences/Graduate Program In Pharmaceutical Sciences
Curated by ChEMBL
School Of Health Sciences/Graduate Program In Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 845nMAssay Description:Inhibition of human acetylcholinesterase using acetylthiocholine iodide as substrate incubated for 15 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
School Of Health Sciences/Graduate Program In Pharmaceutical Sciences
Curated by ChEMBL
School Of Health Sciences/Graduate Program In Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 903nMAssay Description:Inhibition of human acetylcholinesterase using acetylthiocholine iodide as substrate incubated for 15 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
School Of Health Sciences/Graduate Program In Pharmaceutical Sciences
Curated by ChEMBL
School Of Health Sciences/Graduate Program In Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 912nMAssay Description:Inhibition of human acetylcholinesterase using acetylthiocholine iodide as substrate incubated for 15 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
School Of Health Sciences/Graduate Program In Pharmaceutical Sciences
Curated by ChEMBL
School Of Health Sciences/Graduate Program In Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 988nMAssay Description:Inhibition of human acetylcholinesterase using acetylthiocholine iodide as substrate incubated for 15 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of HIV1 integrase strand transfer activityMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of HIV1 integrase 3'-end processing activityMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of HIV1 integrase 3'-end processing activityMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of HIV1 integrase strand transfer activityMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of HIV1 integrase 3'-end processing activityMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of HIV1 integrase strand transfer activityMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of HIV1 integrase strand transfer activityMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
School Of Health Sciences/Graduate Program In Pharmaceutical Sciences
Curated by ChEMBL
School Of Health Sciences/Graduate Program In Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 5.64E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of HIV1 integrase 3'-end processing activityMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
School Of Health Sciences/Graduate Program In Pharmaceutical Sciences
Curated by ChEMBL
School Of Health Sciences/Graduate Program In Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 6.99E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of HIV1 integrase 3'-end processing activityMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
School Of Health Sciences/Graduate Program In Pharmaceutical Sciences
Curated by ChEMBL
School Of Health Sciences/Graduate Program In Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 7.34E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PTPA after 20 mins by ELISAMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant protein tyrosine phosphataseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
School Of Health Sciences/Graduate Program In Pharmaceutical Sciences
Curated by ChEMBL
School Of Health Sciences/Graduate Program In Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 8.74E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis)
Universidade Federal De Santa Catarina
Curated by ChEMBL
Universidade Federal De Santa Catarina
Curated by ChEMBL
Affinity DataIC50: 8.80E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis PTP-AMore data for this Ligand-Target Pair