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Found 258 with Last Name = 'zong' and Initial = 'x'
TargetEndothelin-1 receptor(RAT)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50064000(CHEMBL3400988)
Affinity DataIC50:  3.30nMAssay Description:Displacement of PD156707 from rat ETA receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50063998(CHEMBL3400989)
Affinity DataIC50:  3.90nMAssay Description:Displacement of [125I]ET-1 from rat ETA receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50061101(4-(1,1-Dimethylethyl)-N-(6-(2-hydroxyethoxy)-5-(2-...)
Affinity DataIC50:  4.70nMAssay Description:Displacement of [125I]ET-1 from rat ETA receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50063997(CHEMBL3400996)
Affinity DataIC50:  5.5nMAssay Description:Displacement of [125I]ET-1 from rat ETA receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50063999(CHEMBL3400984)
Affinity DataIC50:  12nMAssay Description:Displacement of [125I]ET-1 from rat ETA receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50063996(CHEMBL3400998)
Affinity DataIC50:  19nMAssay Description:Displacement of [125I]ET-1 from rat ETA receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnoctamin-1(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50594075(CHEMBL5186789)
Affinity DataIC50:  24nMAssay Description:Inhibition of YFP tagged ANO1 (unknown origin) expressed in FRT cells incubated for 24 hrs by fluorescence plate reader assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAnoctamin-1(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM11242(5-chloro-N-(2-chloro-4-nitrophenyl)-2-hydroxybenza...)
Affinity DataIC50:  28nMAssay Description:Inhibition of YFP tagged ANO1 (unknown origin) expressed in FRT cells incubated for 24 hrs by fluorescence plate reader assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetEndothelin-1 receptor(RAT)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50029352(CHEMBL336033 | [(5S,8S,11R,14S,16aR)-8-(1H-Indol-3...)
Affinity DataIC50:  28nMAssay Description:Displacement of [125I]ET-1 from rat ETA receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnoctamin-1(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50594073(CHEMBL5206041)
Affinity DataIC50:  29nMAssay Description:Inhibition of YFP tagged ANO1 (unknown origin) expressed in FRT cells incubated for 24 hrs by fluorescence plate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAnoctamin-1(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50239459(CHEMBL4074929)
Affinity DataIC50:  30nMAssay Description:Inhibition of YFP tagged ANO1 (unknown origin) expressed in FRT cells incubated for 24 hrs by fluorescence plate reader assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50082211(CHEMBL3421742)
Affinity DataIC50:  60nMAssay Description:Inhibition of recombinant HDAC1 (unknown origin) using fluorogenic substrate Boc-Lys (acetyl)-AMC after 20 mins by homogeneous fluorescence release a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50029422(CHEMBL3343311)
Affinity DataIC50:  61nMAssay Description:Inhibition of Aurora-A (unknown origin) using STK substrate 2-biotin by HTRF-KinEASE-STK assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50082261(CHEMBL3421746)
Affinity DataIC50:  70nMAssay Description:Inhibition of recombinant HDAC1 (unknown origin) using fluorogenic substrate Boc-Lys (acetyl)-AMC after 20 mins by homogeneous fluorescence release a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50094049(CHEMBL3585965)
Affinity DataIC50:  70nMAssay Description:Inhibition of recombinant HDAC1 (unknown origin) incubated for 10 mins using Boc-Lys(acetyl)-AMC fluorogenic substrate by homogeneous fluorescence re...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50029416(CHEMBL3343310)
Affinity DataIC50:  78nMAssay Description:Inhibition of Aurora-A (unknown origin) using STK substrate 2-biotin by HTRF-KinEASE-STK assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50094054(CHEMBL3585968)
Affinity DataIC50:  80nMAssay Description:Inhibition of recombinant HDAC1 (unknown origin) incubated for 10 mins using Boc-Lys(acetyl)-AMC fluorogenic substrate by homogeneous fluorescence re...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50029449(CHEMBL3343321)
Affinity DataIC50:  82nMAssay Description:Inhibition of Aurora-A (unknown origin) using STK substrate 2-biotin by HTRF-KinEASE-STK assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50082210(CHEMBL3421741)
Affinity DataIC50:  90nMAssay Description:Inhibition of recombinant HDAC1 (unknown origin) using fluorogenic substrate Boc-Lys (acetyl)-AMC after 20 mins by homogeneous fluorescence release a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50061101(4-(1,1-Dimethylethyl)-N-(6-(2-hydroxyethoxy)-5-(2-...)
Affinity DataIC50:  95nMAssay Description:Displacement of [125I]ET-1 from rat ETB receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50029447(CHEMBL3343320)
Affinity DataIC50:  103nMAssay Description:Inhibition of Aurora-A (unknown origin) using STK substrate 2-biotin by HTRF-KinEASE-STK assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50082213(CHEMBL3421743)
Affinity DataIC50:  110nMAssay Description:Inhibition of recombinant HDAC1 (unknown origin) using fluorogenic substrate Boc-Lys (acetyl)-AMC after 20 mins by homogeneous fluorescence release a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50029459(CHEMBL3343420)
Affinity DataIC50:  110nMAssay Description:Inhibition of Aurora-A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50029454(CHEMBL3343418)
Affinity DataIC50:  115nMAssay Description:Inhibition of Aurora-A (unknown origin) using STK substrate 2-biotin by HTRF-KinEASE-STK assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50094053(CHEMBL3585967)
Affinity DataIC50:  120nMAssay Description:Inhibition of recombinant HDAC1 (unknown origin) incubated for 10 mins using Boc-Lys(acetyl)-AMC fluorogenic substrate by homogeneous fluorescence re...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50029455(CHEMBL3343419)
Affinity DataIC50:  123nMAssay Description:Inhibition of Aurora-A (unknown origin) using STK substrate 2-biotin by HTRF-KinEASE-STK assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50029429(CHEMBL3343313)
Affinity DataIC50:  128nMAssay Description:Inhibition of Aurora-A (unknown origin) using STK substrate 2-biotin by HTRF-KinEASE-STK assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50029459(CHEMBL3343420)
Affinity DataIC50:  130nMAssay Description:Inhibition of Aurora-B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50029459(CHEMBL3343420)
Affinity DataIC50:  138nMAssay Description:Inhibition of Aurora-A (unknown origin) using STK substrate 2-biotin by HTRF-KinEASE-STK assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50094061(CHEMBL3585970)
Affinity DataIC50:  140nMAssay Description:Inhibition of recombinant HDAC1 (unknown origin) incubated for 10 mins using Boc-Lys(acetyl)-AMC fluorogenic substrate by homogeneous fluorescence re...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50029425(CHEMBL3343314)
Affinity DataIC50:  143nMAssay Description:Inhibition of Aurora-A (unknown origin) using STK substrate 2-biotin by HTRF-KinEASE-STK assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  150nMAssay Description:Inhibition of recombinant HDAC1 (unknown origin) incubated for 10 mins using Boc-Lys(acetyl)-AMC fluorogenic substrate by homogeneous fluorescence re...More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  150nMAssay Description:Inhibition of recombinant HDAC1 (unknown origin) using fluorogenic substrate Boc-Lys (acetyl)-AMC after 20 mins by homogeneous fluorescence release a...More data for this Ligand-Target Pair
TargetHistone deacetylase 2(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50082211(CHEMBL3421742)
Affinity DataIC50:  150nMAssay Description:Inhibition of recombinant HDAC2 (unknown origin) using fluorogenic substrate Boc-Lys (acetyl)-AMC after 20 mins by homogeneous fluorescence release a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50029459(CHEMBL3343420)
Affinity DataIC50:  156nMAssay Description:Inhibition of Aurora-B (unknown origin) using STK substrate 2-biotin by HTRF-KinEASE-STK assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50029453(CHEMBL3343417)
Affinity DataIC50:  157nMAssay Description:Inhibition of Aurora-A (unknown origin) using STK substrate 2-biotin by HTRF-KinEASE-STK assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50029422(CHEMBL3343311)
Affinity DataIC50:  172nMAssay Description:Inhibition of Aurora-B (unknown origin) using STK substrate 2-biotin by HTRF-KinEASE-STK assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50029455(CHEMBL3343419)
Affinity DataIC50:  176nMAssay Description:Inhibition of Aurora-B (unknown origin) using STK substrate 2-biotin by HTRF-KinEASE-STK assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50082208(CHEMBL3421739)
Affinity DataIC50:  180nMAssay Description:Inhibition of recombinant HDAC1 (unknown origin) using fluorogenic substrate Boc-Lys (acetyl)-AMC after 20 mins by homogeneous fluorescence release a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50029454(CHEMBL3343418)
Affinity DataIC50:  181nMAssay Description:Inhibition of Aurora-B (unknown origin) using STK substrate 2-biotin by HTRF-KinEASE-STK assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50063997(CHEMBL3400996)
Affinity DataIC50:  183nMAssay Description:Displacement of [125I]ET-1 from rat ETB receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50094047(CHEMBL3585964)
Affinity DataIC50:  190nMAssay Description:Inhibition of recombinant HDAC1 (unknown origin) incubated for 10 mins using Boc-Lys(acetyl)-AMC fluorogenic substrate by homogeneous fluorescence re...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50029444(CHEMBL3343318)
Affinity DataIC50:  193nMAssay Description:Inhibition of Aurora-A (unknown origin) using STK substrate 2-biotin by HTRF-KinEASE-STK assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50029416(CHEMBL3343310)
Affinity DataIC50:  193nMAssay Description:Inhibition of Aurora-B (unknown origin) using STK substrate 2-biotin by HTRF-KinEASE-STK assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50029367(CHEMBL3343309)
Affinity DataIC50:  195nMAssay Description:Inhibition of Aurora-A (unknown origin) using STK substrate 2-biotin by HTRF-KinEASE-STK assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50029429(CHEMBL3343313)
Affinity DataIC50:  196nMAssay Description:Inhibition of Aurora-B (unknown origin) using STK substrate 2-biotin by HTRF-KinEASE-STK assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50029449(CHEMBL3343321)
Affinity DataIC50:  197nMAssay Description:Inhibition of Aurora-B (unknown origin) using STK substrate 2-biotin by HTRF-KinEASE-STK assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50063998(CHEMBL3400989)
Affinity DataIC50:  198nMAssay Description:Displacement of [125I]ET-1 from rat ETB receptor after 1 hr by Lowry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50082262(CHEMBL3421747)
Affinity DataIC50:  200nMAssay Description:Inhibition of recombinant HDAC8 (unknown origin) using fluorogenic substrate Boc-Lys (acetyl)-AMC after 20 mins by homogeneous fluorescence release a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50029446(CHEMBL3343319)
Affinity DataIC50:  202nMAssay Description:Inhibition of Aurora-A (unknown origin) using STK substrate 2-biotin by HTRF-KinEASE-STK assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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