TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataKi: 38nMAssay Description:Non-competitive inhibition of Electrophorus electricus AChE using acetylthiocholine iodide as substrate pretreated for 10 mins followed by substrate ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataKi: 1.04E+3nMAssay Description:Inhibition of BRD4 (unknown origin) expressed in human H1299 cells co-expressing HPV16-LCR/E2 after 24 hrs by Bright Glo-luciferase reporter gene ass...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataKi: 2.45E+3nMAssay Description:Non-competitive inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition b...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataKi: 7.76E+3nMAssay Description:Non-competitive inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition b...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataKi: 8.42E+3nMAssay Description:Apparent affinity to inhibit binding of [3H]-pCCK-8 to Cholecystokinin type A receptor of guinea pig pancreatic membranesMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataKi: 8.60E+3nMAssay Description:Non-competitive inhibition of electric eel acetylcholine esterase using acetylcholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataKi: 9.70E+3nMAssay Description:Affinity of compound to Sigma opioid receptor labelled with [3H](+)-3-PPPMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataKi: 1.04E+4nMAssay Description:Non-competitive inhibition of electric eel acetylcholine esterase using acetylcholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataKi: 1.15E+4nMAssay Description:Non-competitive inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition b...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataKi: 1.34E+4nMAssay Description:Non-competitive inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition b...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataKi: 1.70E+4nMAssay Description:Non-competitive inhibition of electric eel acetylcholine esterase using acetylcholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataKi: 1.90E+4nMAssay Description:Non-competitive inhibition of electric eel acetylcholine esterase using acetylcholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataKi: 2.11E+4nMAssay Description:Non-competitive inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition b...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataKi: 2.24E+4nMAssay Description:Non-competitive inhibition of electric eel acetylcholine esterase using acetylcholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataKi: 2.24E+4nMAssay Description:Mixed inhibition of electric eel acetylcholine esterase using acetylcholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataKi: 2.44E+4nMAssay Description:Non-competitive inhibition of electric eel acetylcholine esterase using acetylcholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 5.70nMAssay Description:Apparent affinity to inhibit binding of [3H]-pCCK-8 to Cholecystokinin type A receptor of guinea pig pancreatic membranesMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's metho...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibition of Electrophorus electricus AChE using acetylthiocholine iodide as substrate pretreated for 10 mins followed by substrate addition measure...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universidade Federal Do Abc
Curated by ChEMBL
Universidade Federal Do Abc
Curated by ChEMBL
Affinity DataIC50: 159nMAssay Description:Displacement of fluormone from human PPARgamma LBD expressed in Escherichia coli BL21 DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataIC50: 460nMAssay Description:Inhibition of Electrophorus electricus AChE using acetylthiocholine iodide as substrate pretreated for 10 mins followed by substrate addition measure...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universidade Federal Do Abc
Curated by ChEMBL
Universidade Federal Do Abc
Curated by ChEMBL
Affinity DataIC50: 1.14E+3nMAssay Description:Displacement of fluormone from human PPARgamma LBD expressed in Escherichia coli BL21 DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.01E+3nMAssay Description:Inhibition of human acetylcholine esterase preincubated for 10 mins followed by the addition of 550 uM of acetylcholine iodide as substrate measured ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universidade Federal Do Abc
Curated by ChEMBL
Universidade Federal Do Abc
Curated by ChEMBL
Affinity DataIC50: 2.22E+3nMAssay Description:Displacement of fluormone from human PPARgamma LBD expressed in Escherichia coli BL21 DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataIC50: 2.71E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's metho...More data for this Ligand-Target Pair
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of horse butyrylcholine esterase preincubated for 10 mins followed by the addition of butyrylcholine iodide as substrate measured after 5 ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataIC50: 3.15E+3nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as a substrate incubated for 10 mins by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 4.69E+3nMAssay Description:Binding affinity of [3H]spiroperidol to striatal Dopamine receptor D2 binding sitesMore data for this Ligand-Target Pair
Affinity DataIC50: 4.69E+3nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine iodide as substrate pretreated for 10 mins followed by substrate addition measured at 12 se...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of horse butyrylcholine esterase preincubated for 10 mins followed by the addition of butyrylcholine iodide as substrate measured after 5 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universidade Federal Do Abc
Curated by ChEMBL
Universidade Federal Do Abc
Curated by ChEMBL
Affinity DataIC50: 5.13E+3nMAssay Description:Displacement of fluormone from human PPARgamma LBD expressed in Escherichia coli BL21 DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.65E+3nMAssay Description:Inhibition of human acetylcholine esterase preincubated for 10 mins followed by the addition of 550 uM of acetylcholine iodide as substrate measured ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataIC50: 6.60E+3nMAssay Description:Inhibition of electric eel acetylcholine esterase preincubated for 10 mins followed by the addition of acetylcholine iodide as substrate measured aft...More data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of horse butyrylcholine esterase preincubated for 10 mins followed by the addition of butyrylcholine iodide as substrate measured after 5 ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataIC50: 8.65E+3nMAssay Description:Inhibition activity against AICAR formyltransferase determined against L cellMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataIC50: 1.04E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's metho...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataIC50: 1.09E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's metho...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataIC50: 1.19E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's metho...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataIC50: 1.32E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's metho...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataIC50: 1.37E+4nMAssay Description:Inhibition of electric eel acetylcholine esterase preincubated for 10 mins followed by the addition of acetylcholine iodide as substrate measured aft...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataIC50: 1.43E+4nMAssay Description:Inhibition of electric eel acetylcholine esterase preincubated for 10 mins followed by the addition of acetylcholine iodide as substrate measured aft...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataIC50: 1.47E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's metho...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataIC50: 1.61E+4nMAssay Description:Inhibition of electric eel acetylcholine esterase preincubated for 10 mins followed by the addition of acetylcholine iodide as substrate measured aft...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataIC50: 1.61E+4nMAssay Description:Inhibition of electric eel acetylcholine esterase preincubated for 10 mins followed by the addition of acetylcholine iodide as substrate measured aft...More data for this Ligand-Target Pair
Affinity DataIC50: 1.64E+4nMAssay Description:Inhibition of horse butyrylcholine esterase preincubated for 10 mins followed by the addition of butyrylcholine iodide as substrate measured after 5 ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataIC50: 1.67E+4nMAssay Description:Inhibition of Electrophorus electricus AChE using acetylthiocholine iodide as substrate pretreated for 10 mins followed by substrate addition measure...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataIC50: 1.72E+4nMAssay Description:Inhibition of electric eel acetylcholine esterase preincubated for 10 mins followed by the addition of acetylcholine iodide as substrate measured aft...More data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of horse butyrylcholine esterase preincubated for 10 mins followed by the addition of butyrylcholine iodide as substrate measured after 5 ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataIC50: 1.96E+4nMAssay Description:Inhibition of electric eel acetylcholine esterase preincubated for 10 mins followed by the addition of acetylcholine iodide as substrate measured aft...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas
Curated by ChEMBL
Federal University of Alfenas
Curated by ChEMBL
Affinity DataIC50: 2.15E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's metho...More data for this Ligand-Target Pair