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Found 77 with Last Name = 'da silva' and Initial = 'fm'
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataKi:  38nMAssay Description:Non-competitive inhibition of Electrophorus electricus AChE using acetylthiocholine iodide as substrate pretreated for 10 mins followed by substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM50256407(CHEMBL4088197)
Affinity DataKi:  1.04E+3nMAssay Description:Inhibition of BRD4 (unknown origin) expressed in human H1299 cells co-expressing HPV16-LCR/E2 after 24 hrs by Bright Glo-luciferase reporter gene ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM50292422(CHEMBL4175724)
Affinity DataKi:  2.45E+3nMAssay Description:Non-competitive inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM50292419(CHEMBL4163724)
Affinity DataKi:  7.76E+3nMAssay Description:Non-competitive inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM50292536(CHEMBL4170841)
Affinity DataKi:  8.42E+3nMAssay Description:Apparent affinity to inhibit binding of [3H]-pCCK-8 to Cholecystokinin type A receptor of guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM50139050(CHEMBL3753906)
Affinity DataKi:  8.60E+3nMAssay Description:Non-competitive inhibition of electric eel acetylcholine esterase using acetylcholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM50292510(CHEMBL4172314)
Affinity DataKi:  9.70E+3nMAssay Description:Affinity of compound to Sigma opioid receptor labelled with [3H](+)-3-PPPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM50139006(CHEMBL3753607)
Affinity DataKi:  1.04E+4nMAssay Description:Non-competitive inhibition of electric eel acetylcholine esterase using acetylcholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM50292423(CHEMBL4167867)
Affinity DataKi:  1.15E+4nMAssay Description:Non-competitive inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM50292442(CHEMBL4171226)
Affinity DataKi:  1.34E+4nMAssay Description:Non-competitive inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM50139052(CHEMBL3754700)
Affinity DataKi:  1.70E+4nMAssay Description:Non-competitive inhibition of electric eel acetylcholine esterase using acetylcholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM50139049(CHEMBL3753732)
Affinity DataKi:  1.90E+4nMAssay Description:Non-competitive inhibition of electric eel acetylcholine esterase using acetylcholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM50292526(CHEMBL4164436)
Affinity DataKi:  2.11E+4nMAssay Description:Non-competitive inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM50139051(CHEMBL3753070)
Affinity DataKi:  2.24E+4nMAssay Description:Non-competitive inhibition of electric eel acetylcholine esterase using acetylcholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM50139007(CHEMBL3754287)
Affinity DataKi:  2.24E+4nMAssay Description:Mixed inhibition of electric eel acetylcholine esterase using acetylcholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM50139053(CHEMBL3752227)
Affinity DataKi:  2.44E+4nMAssay Description:Non-competitive inhibition of electric eel acetylcholine esterase using acetylcholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Federal University Of Alfenas

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  5.70nMAssay Description:Apparent affinity to inhibit binding of [3H]-pCCK-8 to Cholecystokinin type A receptor of guinea pig pancreatic membranesMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  26nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  26nMAssay Description:Inhibition of Electrophorus electricus AChE using acetylthiocholine iodide as substrate pretreated for 10 mins followed by substrate addition measure...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50030474(Avandamet | Avandaryl | Avandia | BRL-49653 | CHEB...)
Affinity DataIC50:  159nMAssay Description:Displacement of fluormone from human PPARgamma LBD expressed in Escherichia coli BL21 DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM50256407(CHEMBL4088197)
Affinity DataIC50:  460nMAssay Description:Inhibition of Electrophorus electricus AChE using acetylthiocholine iodide as substrate pretreated for 10 mins followed by substrate addition measure...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM53804(4-({2-[(1,3-dioxo-1,3-dihydro-2H-inden-2-ylidene)m...)
Affinity DataIC50:  1.14E+3nMAssay Description:Displacement of fluormone from human PPARgamma LBD expressed in Escherichia coli BL21 DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Federal University Of Alfenas

Curated by ChEMBL
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  2.01E+3nMAssay Description:Inhibition of human acetylcholine esterase preincubated for 10 mins followed by the addition of 550 uM of acetylcholine iodide as substrate measured ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50387185(CHEMBL2048021)
Affinity DataIC50:  2.22E+3nMAssay Description:Displacement of fluormone from human PPARgamma LBD expressed in Escherichia coli BL21 DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM50292422(CHEMBL4175724)
Affinity DataIC50:  2.71E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139052(CHEMBL3754700)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of horse butyrylcholine esterase preincubated for 10 mins followed by the addition of butyrylcholine iodide as substrate measured after 5 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM50590393(CHEMBL5195581)
Affinity DataIC50:  3.15E+3nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as a substrate incubated for 10 mins by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  4.69E+3nMAssay Description:Binding affinity of [3H]spiroperidol to striatal Dopamine receptor D2 binding sitesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  4.69E+3nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine iodide as substrate pretreated for 10 mins followed by substrate addition measured at 12 se...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139053(CHEMBL3752227)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of horse butyrylcholine esterase preincubated for 10 mins followed by the addition of butyrylcholine iodide as substrate measured after 5 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universidade Federal Do Abc

Curated by ChEMBL
LigandPNGBDBM50493700(CHEMBL1426715)
Affinity DataIC50:  5.13E+3nMAssay Description:Displacement of fluormone from human PPARgamma LBD expressed in Escherichia coli BL21 DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Federal University Of Alfenas

Curated by ChEMBL
LigandPNGBDBM50139053(CHEMBL3752227)
Affinity DataIC50:  5.65E+3nMAssay Description:Inhibition of human acetylcholine esterase preincubated for 10 mins followed by the addition of 550 uM of acetylcholine iodide as substrate measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM50139053(CHEMBL3752227)
Affinity DataIC50:  6.60E+3nMAssay Description:Inhibition of electric eel acetylcholine esterase preincubated for 10 mins followed by the addition of acetylcholine iodide as substrate measured aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139006(CHEMBL3753607)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of horse butyrylcholine esterase preincubated for 10 mins followed by the addition of butyrylcholine iodide as substrate measured after 5 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM50292442(CHEMBL4171226)
Affinity DataIC50:  8.65E+3nMAssay Description:Inhibition activity against AICAR formyltransferase determined against L cellMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM50292536(CHEMBL4170841)
Affinity DataIC50:  1.04E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM50292510(CHEMBL4172314)
Affinity DataIC50:  1.09E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM50292539(CHEMBL4174394)
Affinity DataIC50:  1.19E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM50292423(CHEMBL4167867)
Affinity DataIC50:  1.32E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM50139050(CHEMBL3753906)
Affinity DataIC50:  1.37E+4nMAssay Description:Inhibition of electric eel acetylcholine esterase preincubated for 10 mins followed by the addition of acetylcholine iodide as substrate measured aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM50139051(CHEMBL3753070)
Affinity DataIC50:  1.43E+4nMAssay Description:Inhibition of electric eel acetylcholine esterase preincubated for 10 mins followed by the addition of acetylcholine iodide as substrate measured aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM50292565(CHEMBL4160612)
Affinity DataIC50:  1.47E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM50139006(CHEMBL3753607)
Affinity DataIC50:  1.61E+4nMAssay Description:Inhibition of electric eel acetylcholine esterase preincubated for 10 mins followed by the addition of acetylcholine iodide as substrate measured aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM50139049(CHEMBL3753732)
Affinity DataIC50:  1.61E+4nMAssay Description:Inhibition of electric eel acetylcholine esterase preincubated for 10 mins followed by the addition of acetylcholine iodide as substrate measured aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139007(CHEMBL3754287)
Affinity DataIC50:  1.64E+4nMAssay Description:Inhibition of horse butyrylcholine esterase preincubated for 10 mins followed by the addition of butyrylcholine iodide as substrate measured after 5 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM50256425(CHEMBL4066925)
Affinity DataIC50:  1.67E+4nMAssay Description:Inhibition of Electrophorus electricus AChE using acetylthiocholine iodide as substrate pretreated for 10 mins followed by substrate addition measure...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM50139052(CHEMBL3754700)
Affinity DataIC50:  1.72E+4nMAssay Description:Inhibition of electric eel acetylcholine esterase preincubated for 10 mins followed by the addition of acetylcholine iodide as substrate measured aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139049(CHEMBL3753732)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of horse butyrylcholine esterase preincubated for 10 mins followed by the addition of butyrylcholine iodide as substrate measured after 5 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM50139007(CHEMBL3754287)
Affinity DataIC50:  1.96E+4nMAssay Description:Inhibition of electric eel acetylcholine esterase preincubated for 10 mins followed by the addition of acetylcholine iodide as substrate measured aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Federal University of Alfenas

Curated by ChEMBL
LigandPNGBDBM50292566(CHEMBL4168953)
Affinity DataIC50:  2.15E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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