Affinity DataKi: 0.200nMAssay Description:In vitro inhibitory constant against [3H]-paroxetine binding to rat frontal cortex membrane serotonin reuptake siteMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:In vitro inhibitory constant against [3H]-paroxetine binding to rat frontal cortex membrane serotonin reuptake siteMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:In vitro inhibitory constant against [3H]-paroxetine binding to rat frontal cortex membrane serotonin reuptake siteMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:In vitro inhibitory constant against [3H]-paroxetine binding to rat frontal cortex membrane serotonin reuptake siteMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:In vitro inhibitory constant against [3H]-paroxetine binding to rat frontal cortex membrane serotonin reuptake siteMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:In vitro inhibitory constant against [3H]-paroxetine binding to rat frontal cortex membrane serotonin reuptake siteMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:In vitro inhibitory constant against [3H]-paroxetine binding to rat frontal cortex membrane serotonin reuptake siteMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:In vitro inhibitory constant against [3H]-paroxetine binding to rat frontal cortex membrane serotonin reuptake siteMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:In vitro inhibitory constant against [3H]-paroxetine binding to rat frontal cortex membrane serotonin reuptake siteMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:In vitro inhibitory constant against [3H]-paroxetine binding to rat frontal cortex membrane serotonin reuptake siteMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:In vitro inhibitory constant against [3H]-paroxetine binding to rat frontal cortex membrane serotonin reuptake siteMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:In vitro inhibitory constant against [3H]-paroxetine binding to rat frontal cortex membrane serotonin reuptake siteMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:In vitro inhibitory constant against [3H]-spiperone binding to human dopamine D2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:In vitro inhibitory constant against [3H]-spiperone binding to human dopamine D2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.03nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:In vitro inhibitory constant against [3H]-paroxetine binding to rat frontal cortex membrane serotonin reuptake siteMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:In vitro inhibitory constant against [3H]-paroxetine binding to rat frontal cortex membrane serotonin reuptake siteMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:In vitro inhibitory constant against [3H]-paroxetine binding to rat frontal cortex membrane serotonin reuptake siteMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:In vitro inhibitory constant against [3H]-paroxetine binding to rat frontal cortex membrane serotonin reuptake siteMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products
Curated by ChEMBL
Abbott Healthcare Products
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]-N-Methyl-Lysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:In vitro inhibitory constant against [3H]-paroxetine binding to rat frontal cortex membrane serotonin reuptake siteMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:In vitro inhibitory constant against [3H]-paroxetine binding to rat frontal cortex membrane serotonin reuptake siteMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:In vitro inhibitory constant against [3H]-paroxetine binding to rat frontal cortex membrane serotonin reuptake siteMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products
Curated by ChEMBL
Abbott Healthcare Products
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]-N-Methyl-Lysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:In vitro inhibitory constant against [3H]-paroxetine binding to rat frontal cortex membrane serotonin reuptake siteMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:In vitro inhibitory constant against [3H]-spiperone binding to human dopamine D2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [3H]CP-55940 from human cannabinoid CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:In vitro inhibitory constant against [3H]-paroxetine binding to rat frontal cortex membrane serotonin reuptake siteMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:In vitro inhibitory constant against [3H]-spiperone binding to human dopamine D2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:In vitro inhibitory constant against [3H]-paroxetine binding to rat frontal cortex membrane serotonin reuptake siteMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:In vitro inhibitory constant against [3H]-paroxetine binding to rat frontal cortex membrane serotonin reuptake siteMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:In vitro inhibitory constant against [3H]-paroxetine binding to rat frontal cortex membrane serotonin reuptake siteMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:In vitro inhibitory constant against [3H]-paroxetine binding to rat frontal cortex membrane serotonin reuptake siteMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:In vitro inhibitory constant against [3H]-spiperone binding to human dopamine D2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:In vitro inhibitory constant against [3H]-spiperone binding to human dopamine D2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Displacement of [3H]CP-55940 from human cannabinoid CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:In vitro inhibitory constant against [3H]-spiperone binding to human dopamine D2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products
Curated by ChEMBL
Abbott Healthcare Products
Curated by ChEMBL
Affinity DataKi: 4.80nMAssay Description:Displacement of [3H]-N-Methyl-Lysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:In vitro inhibitory constant against [3H]-spiperone binding to human dopamine D2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:In vitro inhibitory constant against [3H]-spiperone binding to human dopamine D2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products
Curated by ChEMBL
Abbott Healthcare Products
Curated by ChEMBL
Affinity DataKi: 5.80nMAssay Description:Displacement of [3H]-N-Methyl-Lysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation count...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products
Curated by ChEMBL
Abbott Healthcare Products
Curated by ChEMBL
Affinity DataKi: 6.10nMAssay Description:Displacement of [3H]-N-Methyl-Lysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 6.90nMAssay Description:In vitro inhibitory constant against [3H]-spiperone binding to human dopamine D2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Solvay Pharmaceuticals
Curated by PDSP Ki Database
Solvay Pharmaceuticals
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products
Curated by ChEMBL
Abbott Healthcare Products
Curated by ChEMBL
Affinity DataKi: 7.10nMAssay Description:Displacement of [3H]-N-Methyl-Lysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation count...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products
Curated by ChEMBL
Abbott Healthcare Products
Curated by ChEMBL
Affinity DataKi: 7.20nMAssay Description:Displacement of [3H]-N-Methyl-Lysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation count...More data for this Ligand-Target Pair