Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetProbable G-protein coupled receptor 139(Homo sapiens (Human))
Takeda California

Curated by ChEMBL

LigandBDBM50566752(CHEMBL4874147)Copy SMILESCopy InChI

Affinity DataKi:  1.16E+3nMAssay Description:Displacement of (S)-N-(1-(2-[3H]-4-methoxyphenyl)propan-2-yl)-2-(2,3-dimethyl-7-oxothieno[2,3-d]pyridazin-6(7H)-yl)acetamide from human GPR139 expres...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetProbable G-protein coupled receptor 139(Homo sapiens (Human))
Takeda California

Curated by ChEMBL

LigandBDBM50566752(CHEMBL4874147)Copy SMILESCopy InChI

Affinity DataEC50:  33nMAssay Description:Agonist activity at human GPR139 expressed in CHO-TRex cells assessed as stimulation of calcium signalling incubated for 15 mins by FLIPR assayMore data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI