Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetDNA gyrase subunit A(Escherichia coli (strain K12))
Astrazeneca

US Patent
LigandPNGBDBM139376(US8889671, 5)
Affinity DataIC50:  169nMpH: 7.5Assay Description:In a black, 384-well polystyrene assay plate, 30 microliters/well of 5 nM Escherichia coli DNA gyrase A/B tetramer and 130 micrograms/mL of topologic...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDNA gyrase subunit A/B(Staphylococcus aureus)
University Of Cape Town

Curated by ChEMBL
LigandPNGBDBM139376(US8889671, 5)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of Staphylococcus aureus ATTC 25923 DNA gyraseMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDNA gyrase subunit B(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University Of Cape Town

Curated by ChEMBL
LigandPNGBDBM139376(US8889671, 5)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv DNA gyraseMore data for this Ligand-Target Pair
In DepthDetails PubMed