Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetCholine kinase(Plasmodium falciparum (isolate 3D7))
Universidad De Granada

Curated by ChEMBL
LigandPNGBDBM50166172(Bisquinolinium derivative | CHEMBL192986)
Affinity DataIC50:  1.75E+3nMAssay Description:Inhibition of Plasmodium falciparum 3D7 choline kinase expressed in Escherichia coli BL21(DE3) assessed as reduction in phosphocholine formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholine kinase alpha(Homo sapiens (Human))
Universidad De Granada

Curated by ChEMBL
LigandPNGBDBM50166172(Bisquinolinium derivative | CHEMBL192986)
Affinity DataIC50:  1.92E+3nMAssay Description:Inhibition of human choline kinase alpha1 using [methyl-14C]choline as substrate assessed as reduction in rate of incorporation of 14C from [methyl-1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholine kinase alpha(Homo sapiens (Human))
Universidad De Granada

Curated by ChEMBL
LigandPNGBDBM50166172(Bisquinolinium derivative | CHEMBL192986)
Affinity DataIC50:  2.00E+3nMAssay Description:Ex vivo inhibitory concentration against human choline kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed