Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 19 hits in this display
BDBM50200384(CHEMBL3968533 | US9763922, Example 299)
BDBM50200384(CHEMBL3968533 | US9763922, Example 299)
IC50: 30nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
BDBM50200384(CHEMBL3968533 | US9763922, Example 299)
BDBM50200384(CHEMBL3968533 | US9763922, Example 299)
BDBM50200384(CHEMBL3968533 | US9763922, Example 299)
BDBM50200384(CHEMBL3968533 | US9763922, Example 299)
IC50: 1.20E+4nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged TAF1 bromodomain 2 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
BDBM50200384(CHEMBL3968533 | US9763922, Example 299)
IC50: 1.30E+4nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged BRD4 bromodomain-1 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
BDBM50200384(CHEMBL3968533 | US9763922, Example 299)
IC50: >2.00E+4nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged TAF1 bromodomain 1 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
BDBM50200384(CHEMBL3968533 | US9763922, Example 299)
IC50: >2.00E+4nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CECR2 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
BDBM50200384(CHEMBL3968533 | US9763922, Example 299)
IC50: >2.00E+4nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged BRD9 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
BDBM50200384(CHEMBL3968533 | US9763922, Example 299)
IC50: >2.00E+4nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged BAZ2B (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
BDBM50200384(CHEMBL3968533 | US9763922, Example 299)
IC50: >2.00E+4nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged BRPF1 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
BDBM50200384(CHEMBL3968533 | US9763922, Example 299)
IC50: >2.00E+4nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged BPTF (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
BDBM50200384(CHEMBL3968533 | US9763922, Example 299)
IC50: >2.00E+4nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged PCAF (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
BDBM50200384(CHEMBL3968533 | US9763922, Example 299)
IC50: >2.00E+4nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged BRD8 bromodomain-1 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
BDBM50200384(CHEMBL3968533 | US9763922, Example 299)
IC50: >2.00E+4nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged BRD4 bromodomain-1 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
BDBM50200384(CHEMBL3968533 | US9763922, Example 299)
IC50: >2.00E+4nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged GCN5 long isoform (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
BDBM50200384(CHEMBL3968533 | US9763922, Example 299)
EC50: 69nMAssay Description:Inhibition of CBP/EP300 in human MOLM16 cells assessed as decrease in MYC expression measured after 4 hrs by RT-PCR analysisMore data for this Ligand-Target Pair
BDBM50200384(CHEMBL3968533 | US9763922, Example 299)
EC50: 910nMAssay Description:Inhibition of CBP/EP300 in human MV4-11 cells assessed as inhibition of MYC expression measured after 4 hrs by luminescence analysisMore data for this Ligand-Target Pair