Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 6 hits in this display
BDBM50326957(4-(5-Chloro-2,3-dihydrobenzofuran-7-yl)-1,1,1-trif...)
BDBM50326957(4-(5-Chloro-2,3-dihydrobenzofuran-7-yl)-1,1,1-trif...)
IC50: 17nMAssay Description:Transrepression activity at glucocorticoid receptor in HFF assessed as inhibition of IL-1-induced IL-6 production after 18 to 24 hrs by ELISAMore data for this Ligand-Target Pair
BDBM50326957(4-(5-Chloro-2,3-dihydrobenzofuran-7-yl)-1,1,1-trif...)
BDBM50326957(4-(5-Chloro-2,3-dihydrobenzofuran-7-yl)-1,1,1-trif...)
BDBM50326957(4-(5-Chloro-2,3-dihydrobenzofuran-7-yl)-1,1,1-trif...)
IC50: >2.00E+3nMAssay Description:Transactivation activity at glucocorticoid receptor in human HeLa cells transfected with luciferase gene linked to MMTV promoter by luciferase assayMore data for this Ligand-Target Pair
BDBM50326957(4-(5-Chloro-2,3-dihydrobenzofuran-7-yl)-1,1,1-trif...)
EC50: 120nMAssay Description:Transactivation activity at glucocorticoid receptor in HFF assessed as induction of aromatase activity after 18 to 24 hrs by ELISAMore data for this Ligand-Target Pair