Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetChymotrypsin-like protease CTRL-1(Homo sapiens (Human))
Centrax International

US Patent
LigandPNGBDBM441781(US10640533, Identification number CX13-137 | US106...)
Affinity DataIC50:  13.5nMAssay Description:Inhibition of the chymotrypsin-like (CT-L), peptidylglutamyl peptide hydrolyzing activity (PGPH), and trypsin-like (T-L) activities of the 20S protea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetChymotrypsin-like protease CTRL-1(Homo sapiens (Human))
Centrax International

US Patent
LigandPNGBDBM441781(US10640533, Identification number CX13-137 | US106...)
Affinity DataIC50:  60.4nMAssay Description:Inhibition of the chymotrypsin-like (CT-L), peptidylglutamyl peptide hydrolyzing activity (PGPH), and trypsin-like (T-L) activities of the 20S protea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
Centrax International

US Patent
LigandPNGBDBM441781(US10640533, Identification number CX13-137 | US106...)
Affinity DataIC50:  5.86E+3nMAssay Description:Inhibition of the chymotrypsin-like (CT-L), peptidylglutamyl peptide hydrolyzing activity (PGPH), and trypsin-like (T-L) activities of the 20S protea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
Centrax International

US Patent
LigandPNGBDBM441781(US10640533, Identification number CX13-137 | US106...)
Affinity DataIC50:  1.19E+4nMAssay Description:Inhibition of the chymotrypsin-like (CT-L), peptidylglutamyl peptide hydrolyzing activity (PGPH), and trypsin-like (T-L) activities of the 20S protea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Centrax International

US Patent
LigandPNGBDBM441781(US10640533, Identification number CX13-137 | US106...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of the chymotrypsin-like (CT-L), peptidylglutamyl peptide hydrolyzing activity (PGPH), and trypsin-like (T-L) activities of the 20S protea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Centrax International

US Patent
LigandPNGBDBM441781(US10640533, Identification number CX13-137 | US106...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of the chymotrypsin-like (CT-L), peptidylglutamyl peptide hydrolyzing activity (PGPH), and trypsin-like (T-L) activities of the 20S protea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent