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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
24
hits in this display
Target
Proteasome subunit beta type-10
(Homo sapiens (Human))
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50529640
(CHEMBL4452892)
Copy SMILES
Copy InChI
Affinity Data
IC50: 71nM
Assay Description:
Inhibition of MECL1 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-10
(Homo sapiens (Human))
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50529640
(CHEMBL4452892)
Copy SMILES
Copy InChI
Affinity Data
IC50: 71nM
Assay Description:
Inhibition of MECL1 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-10
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50529640
(CHEMBL4452892)
Copy SMILES
Copy InChI
Affinity Data
IC50: 305nM
Assay Description:
Inhibition of MECL1 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-10
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50529640
(CHEMBL4452892)
Copy SMILES
Copy InChI
Affinity Data
IC50: 305nM
Assay Description:
Inhibition of MECL1 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-8
(Homo sapiens (Human))
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50529640
(CHEMBL4452892)
Copy SMILES
Copy InChI
Affinity Data
IC50: 346nM
Assay Description:
Inhibition of LMP7 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-8
(Homo sapiens (Human))
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50529640
(CHEMBL4452892)
Copy SMILES
Copy InChI
Affinity Data
IC50: 346nM
Assay Description:
Inhibition of LMP7 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-5
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50529640
(CHEMBL4452892)
Copy SMILES
Copy InChI
Affinity Data
IC50: 378nM
Assay Description:
Inhibition of 20S proteosome beta 5 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-5
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50529640
(CHEMBL4452892)
Copy SMILES
Copy InChI
Affinity Data
IC50: 378nM
Assay Description:
Inhibition of 20S proteosome beta 5 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-2
(Homo sapiens (Human))
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50529640
(CHEMBL4452892)
Copy SMILES
Copy InChI
Affinity Data
IC50: 413nM
Assay Description:
Inhibition of 20S proteosome beta 2 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-2
(Homo sapiens (Human))
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50529640
(CHEMBL4452892)
Copy SMILES
Copy InChI
Affinity Data
IC50: 413nM
Assay Description:
Inhibition of 20S proteosome beta 2 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-5
(Homo sapiens (Human))
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50529640
(CHEMBL4452892)
Copy SMILES
Copy InChI
Affinity Data
IC50: 486nM
Assay Description:
Inhibition of 20S proteosome beta 5 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-5
(Homo sapiens (Human))
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50529640
(CHEMBL4452892)
Copy SMILES
Copy InChI
Affinity Data
IC50: 486nM
Assay Description:
Inhibition of 20S proteosome beta 5 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-2
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50529640
(CHEMBL4452892)
Copy SMILES
Copy InChI
Affinity Data
IC50: 573nM
Assay Description:
Inhibition of 20S proteosome beta 2 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-2
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50529640
(CHEMBL4452892)
Copy SMILES
Copy InChI
Affinity Data
IC50: 573nM
Assay Description:
Inhibition of 20S proteosome beta 2 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-8
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50529640
(CHEMBL4452892)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.92E+3nM
Assay Description:
Inhibition of LMP7 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-8
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50529640
(CHEMBL4452892)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.92E+3nM
Assay Description:
Inhibition of LMP7 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-9
(Homo sapiens (Human))
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50529640
(CHEMBL4452892)
Copy SMILES
Copy InChI
Affinity Data
IC50: >2.50E+4nM
Assay Description:
Inhibition of LMP2 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-1
(Homo sapiens (Human))
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50529640
(CHEMBL4452892)
Copy SMILES
Copy InChI
Affinity Data
IC50: >2.50E+4nM
Assay Description:
Inhibition of 20S proteosome beta 1 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-1
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50529640
(CHEMBL4452892)
Copy SMILES
Copy InChI
Affinity Data
IC50: >2.50E+4nM
Assay Description:
Inhibition of 20S proteosome beta 1 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-1
(Homo sapiens (Human))
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50529640
(CHEMBL4452892)
Copy SMILES
Copy InChI
Affinity Data
IC50: >2.50E+4nM
Assay Description:
Inhibition of 20S proteosome beta 1 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-9
(Homo sapiens (Human))
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50529640
(CHEMBL4452892)
Copy SMILES
Copy InChI
Affinity Data
IC50: >2.50E+4nM
Assay Description:
Inhibition of LMP2 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-1
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50529640
(CHEMBL4452892)
Copy SMILES
Copy InChI
Affinity Data
IC50: >2.50E+4nM
Assay Description:
Inhibition of 20S proteosome beta 1 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-9
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50529640
(CHEMBL4452892)
Copy SMILES
Copy InChI
Affinity Data
IC50: >2.50E+4nM
Assay Description:
Inhibition of LMP2 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-9
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50529640
(CHEMBL4452892)
Copy SMILES
Copy InChI
Affinity Data
IC50: >2.50E+4nM
Assay Description:
Inhibition of LMP2 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI