Home
About
Info
Download
WebServices
Contact
Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
A5LHX3/O14818/P20618/P25786/P25787/P25788/P25789/P28062/P28065/P28066/P28070/P28072/P28074/P40306/P49720/P49721/P60900/Q8TAA3/Q99436
(Homo sapiens (Human))
Cephalon
Curated by
ChEMBL
Ligand
BDBM50031442
(1N-[4-amino(nitroimino)methylamino-1-(1-formyl-3-m...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 2nM
Assay Description:
Compound was evaluated for inhibitory activity against 20S proteasome from human liver and brain
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
antibodypedia
antibodypedia
antibodypedia
antibodypedia
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Patents
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Chymotrypsin-like protease CTRL-1
(Homo sapiens (Human))
TBA
Curated by
ChEMBL
Ligand
BDBM50031442
(1N-[4-amino(nitroimino)methylamino-1-(1-formyl-3-m...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 2nM
Assay Description:
Compound was tested for inhibition of chymotrypsin-like protease of proteasome from postmortem human liver and brain
More data for this Ligand-Target Pair
Target Info
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Patents
In Depth
Details
Article
Copy BDB DOI