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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetProtein-arginine deiminase type-4(Homo sapiens (Human))
University of Toronto

Curated by ChEMBL
LigandPNGBDBM454165(BDBM50246195 | US10716791, Code KP-289)
Affinity DataKi:  4.88E+5nMAssay Description:Inhibition of full length human GST-tagged PAD4 expressed in baculovirus infected Sf9 insect cells preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-4(Homo sapiens (Human))
University of Toronto

Curated by ChEMBL
LigandPNGBDBM454165(BDBM50246195 | US10716791, Code KP-289)
Affinity DataKi:  4.88E+5nMAssay Description:Materials: PAD1, PAD2, PAD3 and PAD4 were purchased from commercial sources. Assay buffer: 50 mM Tris pH 7.5, 100 mM NaCl, 10 mM CaCl2, 5 mM DTT. Col...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-arginine deiminase type-2(Mus musculus)
University Health Network

US Patent
LigandPNGBDBM454165(BDBM50246195 | US10716791, Code KP-289)
Affinity DataKi:  1.79E+6nMAssay Description:Materials: PAD1, PAD2, PAD3 and PAD4 were purchased from commercial sources. Assay buffer: 50 mM Tris pH 7.5, 100 mM NaCl, 10 mM CaCl2, 5 mM DTT. Col...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-arginine deiminase type-2(Mus musculus)
University Health Network

US Patent
LigandPNGBDBM454165(BDBM50246195 | US10716791, Code KP-289)
Affinity DataKi:  1.84E+6nMAssay Description:Inhibition of full length mouse GST-tagged PAD2 expressed in baculovirus infected Sf9 insect cells preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed