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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

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TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM282814(6-((S)-2-Methyl-pyrrolidine-1-carbonyl)-3,4-dihydr...)
Affinity DataIC50:  13nMT: 2°CAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent