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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 12 hits in this display   

TargetPlasminogen(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518241(CHEMBL4569923)
Affinity DataKi:  0.0410nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518241(CHEMBL4569923)
Affinity DataKi:  28nMAssay Description:Inhibition of bovine cationic trypsin using Bz-FVR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518241(CHEMBL4569923)
Affinity DataKi:  1.30E+4nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518241(CHEMBL4569923)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of uPA (unknown origin) using Z-Pyr-Gly-Arg-MCA as substrate after 30 mins relative to untreated controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasma kallikrein(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518241(CHEMBL4569923)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of plasma KLK (unknown origin) using Ac-NLTR-pNA as substrate after 30 mins relative to untreated controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCoagulation factor IX(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518241(CHEMBL4569923)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of activated beta-factor 9 (unknown origin) using Boc-QGR-MCA as substrate after 30 mins relative to untreated controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518241(CHEMBL4569923)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of tPA (unknown origin) using Z-Pyr-Gly-Arg-MCA as substrate after 30 mins relative to untreated controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCoagulation factor XII(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518241(CHEMBL4569923)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of activated beta-factor 12 (unknown origin) using Ac-QRFR-pNA as substrate after 30 mins relative to untreated controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518241(CHEMBL4569923)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of matriptase (unknown origin) using Boc-QAR-MCA as substrate after 30 mins relative to untreated controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518241(CHEMBL4569923)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of activated factor 10 (unknown origin) using Ac-QRSR-pNA as substrate after 30 mins relative to untreated controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCoagulation factor XI(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518241(CHEMBL4569923)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of activated beta-factor 11 (unknown origin) using Bz-FVRpNA as substrate after 30 mins relative to untreated controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518241(CHEMBL4569923)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human thrombin using Ac-ATPR-pNA as substrate after 30 mins relative to untreated controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed