Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetMAP/microtubule affinity-regulating kinase 3(Homo sapiens (Human))
Merck

Curated by ChEMBL

LigandBDBM50208920(CHEMBL3884535)Copy SMILESCopy InChI

Affinity DataIC50:  14nMAssay Description:Inhibition of full length human MARK3 using biotin labeled peptide substrate by HTRF based assayMore data for this Ligand-Target Pair

Target InfoPDBMMDBKEGG
UniProtKB/SwissProt
B.MOADantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetMAP/microtubule affinity-regulating kinase 4(Homo sapiens (Human))
Merck

Curated by ChEMBL

LigandBDBM50208920(CHEMBL3884535)Copy SMILESCopy InChI

Affinity DataIC50:  920nMAssay Description:Inhibition of human MARK4 expressed in HEK293T cells coexpressing tau protein assessed as reduction in tau phosphorylation at Ser262 residues by Alph...More data for this Ligand-Target Pair

Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI