Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetMineralocorticoid receptor(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL

LigandBDBM50597087(CHEMBL5181278)Copy SMILESCopy InChI

Affinity DataKi:  163nMAssay Description:Displacement of [3H]-aldosterone from recombinant human mineralocorticoid receptor expressed in baculovirus infected insect cells incubated overnight...More data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails PubMed
Copy BDB DOI

TargetMineralocorticoid receptor(RAT)
Mitsubishi Tanabe Pharma

Curated by ChEMBL

LigandBDBM50597087(CHEMBL5181278)Copy SMILESCopy InChI

Affinity DataKi:  370nMAssay Description:Displacement of [3H]-aldosterone from rat mineralocorticoid receptor incubated overnight by liquid scintillation counting analysisMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails PubMed
Copy BDB DOI

TargetGlucocorticoid receptor(RAT)
Mitsubishi Tanabe Pharma

Curated by ChEMBL

LigandBDBM50597087(CHEMBL5181278)Copy SMILESCopy InChI

Affinity DataKi:  4.32E+4nMAssay Description:Displacement of [3H]-dexamethasone from rat glucocorticoid receptor incubated overnight by liquid scintillation counting analysisMore data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails PubMed
Copy BDB DOI