Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 10 hits in this display
BDBM43221(2-(benzoylcarbamothioylamino)-5,5-dimethyl-4,7-dih...)
BDBM43221(2-(benzoylcarbamothioylamino)-5,5-dimethyl-4,7-dih...)
BDBM43221(2-(benzoylcarbamothioylamino)-5,5-dimethyl-4,7-dih...)
BDBM43221(2-(benzoylcarbamothioylamino)-5,5-dimethyl-4,7-dih...)
EC50: 99.3nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
BDBM43221(2-(benzoylcarbamothioylamino)-5,5-dimethyl-4,7-dih...)
BDBM43221(2-(benzoylcarbamothioylamino)-5,5-dimethyl-4,7-dih...)
BDBM43221(2-(benzoylcarbamothioylamino)-5,5-dimethyl-4,7-dih...)
EC50: 80.6nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
BDBM43221(2-(benzoylcarbamothioylamino)-5,5-dimethyl-4,7-dih...)
BDBM43221(2-(benzoylcarbamothioylamino)-5,5-dimethyl-4,7-dih...)
EC50: 92.0nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
BDBM43221(2-(benzoylcarbamothioylamino)-5,5-dimethyl-4,7-dih...)
EC50: 171nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair