Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetProteasome subunit beta type-1(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50596498(CHEMBL5177192)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of human constitutive proteasome subunit beta type-1 in human erythrocytes using fluorogenic substrate by UV-spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProteasome subunit beta type-10(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50596498(CHEMBL5177192)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of human proteasome subunit beta type-2i using fluorogenic substrate by UV-spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50596498(CHEMBL5177192)
Affinity DataIC50:  4.60E+4nMAssay Description:Inhibition of human constitutive proteasome subunit beta type-5 in human erythrocytes using fluorogenic substrate by UV-spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50596498(CHEMBL5177192)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human constitutive proteasome subunit beta type-2 in human erythrocytes using fluorogenic substrate by UV-spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProteasome subunit beta type-9(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50596498(CHEMBL5177192)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human proteasome subunit beta type-1i in using fluorogenic substrate by UV-spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50596498(CHEMBL5177192)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of human proteasome subunit beta type-5i using fluorogenic substrate by UV-spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed