Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50302798(2-(3-chloro-5-(2-(2,4-dichloro-5-methylphenylsulfo...)
Affinity DataIC50:  4.70nMAssay Description:Antagonist activity at human CRTH2 expressed in CEM cells assessed as inhibition of PGD2-stimulated cell migration after 3 hrs by transwell migration...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50302798(2-(3-chloro-5-(2-(2,4-dichloro-5-methylphenylsulfo...)
Affinity DataIC50:  10nMAssay Description:Displacement of [3H]-PGD2 from human CRTH2 expressed in HEK 293 cells in presence of 0.5% BSA by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50302798(2-(3-chloro-5-(2-(2,4-dichloro-5-methylphenylsulfo...)
Affinity DataIC50:  8.30E+3nMAssay Description:Displacement of [3H]-PGD2 from human DP receptor expressed in HEK 293 cells in presence of 0.5% BSA by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed