Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Zhejiang Ocean University

Curated by ChEMBL
LigandPNGBDBM144277(US8969333, YW3-56)
Affinity DataIC50:  98nMAssay Description:Inhibition of recombinant human PDE4 using histone H3 as substrate by ELISA-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-4(Homo sapiens (Human))
Zhejiang Ocean University

Curated by ChEMBL
LigandPNGBDBM144277(US8969333, YW3-56)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of PAD4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Zhejiang Ocean University

Curated by ChEMBL
LigandPNGBDBM144277(US8969333, YW3-56)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of PDE4 (unknown origin) by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-6(Homo sapiens (Human))
The Penn State Research Foundation

US Patent
LigandPNGBDBM144277(US8969333, YW3-56)
Affinity DataIC50:  3.50E+3nMT: 2°CAssay Description:The inhibition efficacy of PAD4 inhibitors were determined by colorimetric measurement of citrulline generated by PAD4 catalyzed citrullination of BA...More data for this Ligand-Target Pair
In DepthDetails US Patent