Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetCytochrome P450 2C9(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50105824(4,N-Dimethyl-N-(2-phenyl-2H-pyrazol-3-yl)-benzenes...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory effect on human recombinant liver cytochrome P450 2C9 expressed in yeast strainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C18(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50105824(4,N-Dimethyl-N-(2-phenyl-2H-pyrazol-3-yl)-benzenes...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibitory effect on human recombinant liver cytochrome P450 2C18 expressed in yeast strainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50105824(4,N-Dimethyl-N-(2-phenyl-2H-pyrazol-3-yl)-benzenes...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibitory effect on human recombinant liver cytochrome P450 2C19 expressed in yeast strainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C8(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50105824(4,N-Dimethyl-N-(2-phenyl-2H-pyrazol-3-yl)-benzenes...)
Affinity DataIC50:  1.80E+5nMAssay Description:Inhibitory effect on human recombinant liver Cytochrome P450 2C8 expressed in yeast strainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed