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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Receptor-type tyrosine-protein kinase FLT3
(Homo sapiens (Human))
Nerviano Medical Sciences
US Patent
Ligand
BDBM301795
(N-[6-(2-Benzyloxy-ethoxy)-1H-indazol-3-yl]-4-methy...)
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Affinity Data
IC50: <50nM
Assay Description:
i. Enzyme The assay was performed using FLT3 cytoplasmic domain product and purified in house as GST fused protein. The FLT3 protein (1 microM) was p...
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Mast/stem cell growth factor receptor Kit
(Homo sapiens (Human))
Nerviano Medical Sciences
US Patent
Ligand
BDBM301795
(N-[6-(2-Benzyloxy-ethoxy)-1H-indazol-3-yl]-4-methy...)
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Copy InChI
Affinity Data
IC50: 109nM
Assay Description:
i. Enzyme The assay has been performed using KIT cytoplasmic domain product and purified in house as GST fused protein. The KIT protein (4.5 microM) ...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI