Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 7 hits in this display   

TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8851(3-(4-{4-amino-6-[(4-methylpiperazin-1-yl)methyl]th...)
Affinity DataIC50:  589nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8851(3-(4-{4-amino-6-[(4-methylpiperazin-1-yl)methyl]th...)
Affinity DataIC50:  590nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiopoietin-1 receptor(Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM8851(3-(4-{4-amino-6-[(4-methylpiperazin-1-yl)methyl]th...)
Affinity DataIC50:  630nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiopoietin-1 receptor(Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM8851(3-(4-{4-amino-6-[(4-methylpiperazin-1-yl)methyl]th...)
Affinity DataIC50:  631nMAssay Description:Inhibition of Tie2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8851(3-(4-{4-amino-6-[(4-methylpiperazin-1-yl)methyl]th...)
Affinity DataIC50:  794nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8851(3-(4-{4-amino-6-[(4-methylpiperazin-1-yl)methyl]th...)
Affinity DataIC50:  800nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8851(3-(4-{4-amino-6-[(4-methylpiperazin-1-yl)methyl]th...)
Affinity DataIC50:  800nMAssay Description:Inhibition of c-Kit by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed