Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetProteasome subunit alpha type-1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50577134(CHEMBL4877708)
Affinity DataIC50:  3.80nMAssay Description:Inhibition of caspase-like activity of human proteasome beta-1c subunit using SUC-LLE-AMC as flurogenic substrate preincubated for 15 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50577134(CHEMBL4877708)
Affinity DataIC50:  30nMAssay Description:Inhibition of human proteasome subunit beta-5i chymotrypsin like activity using SUC-ANW-AMC as flurogenic substrate preincubated for 15 mins followed...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50577134(CHEMBL4877708)
Affinity DataIC50:  244nMAssay Description:Inhibition of chymotrypsin-like activity of human 20s proteasome beta 5c subunit using suc-WLA-AMC as flurogenic substrate preincubated for 15 mins f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-9(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50577134(CHEMBL4877708)
Affinity DataIC50:  267nMAssay Description:Inhibition of human caspase-like activity of 20s proteasome beta 1i subunit using SUC-PAL-AMC as flurogenic substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-4(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50577134(CHEMBL4877708)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human trypsin-like activity of 20s proteasome beta 2c subunit using SUC-KQL-AMC as flurogenic substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-10(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50577134(CHEMBL4877708)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of human trypsin-like activity of 20s proteasome beta 2i subunit using SUC-VGR-AMC as flurogenic substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed