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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
6
hits in this display
Target
Proteasome subunit alpha type-1
(Homo sapiens (Human))
Zhejiang University
Curated by
ChEMBL
Ligand
BDBM50577134
(CHEMBL4877708)
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Affinity Data
IC50: 3.80nM
Assay Description:
Inhibition of caspase-like activity of human proteasome beta-1c subunit using SUC-LLE-AMC as flurogenic substrate preincubated for 15 mins followed b...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-8
(Homo sapiens (Human))
Zhejiang University
Curated by
ChEMBL
Ligand
BDBM50577134
(CHEMBL4877708)
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Affinity Data
IC50: 30nM
Assay Description:
Inhibition of human proteasome subunit beta-5i chymotrypsin like activity using SUC-ANW-AMC as flurogenic substrate preincubated for 15 mins followed...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-5
(Homo sapiens (Human))
Zhejiang University
Curated by
ChEMBL
Ligand
BDBM50577134
(CHEMBL4877708)
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Affinity Data
IC50: 244nM
Assay Description:
Inhibition of chymotrypsin-like activity of human 20s proteasome beta 5c subunit using suc-WLA-AMC as flurogenic substrate preincubated for 15 mins f...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-9
(Homo sapiens (Human))
Zhejiang University
Curated by
ChEMBL
Ligand
BDBM50577134
(CHEMBL4877708)
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Affinity Data
IC50: 267nM
Assay Description:
Inhibition of human caspase-like activity of 20s proteasome beta 1i subunit using SUC-PAL-AMC as flurogenic substrate preincubated for 15 mins follow...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-4
(Homo sapiens (Human))
Zhejiang University
Curated by
ChEMBL
Ligand
BDBM50577134
(CHEMBL4877708)
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Affinity Data
IC50: 1.60E+3nM
Assay Description:
Inhibition of human trypsin-like activity of 20s proteasome beta 2c subunit using SUC-KQL-AMC as flurogenic substrate preincubated for 15 mins follow...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-10
(Homo sapiens (Human))
Zhejiang University
Curated by
ChEMBL
Ligand
BDBM50577134
(CHEMBL4877708)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.70E+3nM
Assay Description:
Inhibition of human trypsin-like activity of 20s proteasome beta 2i subunit using SUC-VGR-AMC as flurogenic substrate preincubated for 15 mins follow...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI