Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetChymotrypsin-like protease CTRL-1(Homo sapiens (Human))
Centrax International

US Patent
LigandPNGBDBM441783(US10640533, Identification number CX13-501 | US106...)
Affinity DataIC50:  113nMAssay Description:Inhibition of the chymotrypsin-like (CT-L), peptidylglutamyl peptide hydrolyzing activity (PGPH), and trypsin-like (T-L) activities of the 20S protea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetChymotrypsin-like protease CTRL-1(Homo sapiens (Human))
Centrax International

US Patent
LigandPNGBDBM441783(US10640533, Identification number CX13-501 | US106...)
Affinity DataIC50:  392nMAssay Description:Inhibition of the chymotrypsin-like (CT-L), peptidylglutamyl peptide hydrolyzing activity (PGPH), and trypsin-like (T-L) activities of the 20S protea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Centrax International

US Patent
LigandPNGBDBM441783(US10640533, Identification number CX13-501 | US106...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of the chymotrypsin-like (CT-L), peptidylglutamyl peptide hydrolyzing activity (PGPH), and trypsin-like (T-L) activities of the 20S protea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
Centrax International

US Patent
LigandPNGBDBM441783(US10640533, Identification number CX13-501 | US106...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of the chymotrypsin-like (CT-L), peptidylglutamyl peptide hydrolyzing activity (PGPH), and trypsin-like (T-L) activities of the 20S protea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Centrax International

US Patent
LigandPNGBDBM441783(US10640533, Identification number CX13-501 | US106...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of the chymotrypsin-like (CT-L), peptidylglutamyl peptide hydrolyzing activity (PGPH), and trypsin-like (T-L) activities of the 20S protea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTransmembrane protease serine 11D(Homo sapiens (Human))
Centrax International

US Patent
LigandPNGBDBM441783(US10640533, Identification number CX13-501 | US106...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of the chymotrypsin-like (CT-L), peptidylglutamyl peptide hydrolyzing activity (PGPH), and trypsin-like (T-L) activities of the 20S protea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent