Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL

LigandBDBM50302830(2-(4-(2-(2,4-dichlorophenylsulfonamido)-4-(isoprop...)Copy SMILESCopy InChI

Affinity DataIC50:  2nMAssay Description:Displacement of [3H]-PGD2 from human CRTH2 expressed in HEK 293 cells in presence of 0.5% BSA by scintillation countingMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
DrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetProstaglandin D2 receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL

LigandBDBM50302830(2-(4-(2-(2,4-dichlorophenylsulfonamido)-4-(isoprop...)Copy SMILESCopy InChI

Affinity DataIC50:  36nMAssay Description:Displacement of [3H]-PGD2 from human DP receptor expressed in HEK 293 cells in presence of 0.5% BSA by scintillation countingMore data for this Ligand-Target Pair

Target InfoReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI