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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetProtein-arginine deiminase type-4(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM646232((R)-N-((R)-1-(2-(5-((1S,4R,5R)-4- amino-2-azabicyc...)
Affinity DataIC50:  54.9nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-arginine deiminase type-4(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM646324((R)-N-((R)-1-(2-(5-((1S,4R,5R)-4- amino-2-azabicyc...)
Affinity DataIC50:  55.9nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-arginine deiminase type-4(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM646323((S)-N-((R)-1-(2-(5-((1S,4R,5R)-4- amino-2-azabicyc...)
Affinity DataIC50:  67.6nMAssay Description:One hundred nanoliters of test compounds dissolved in DMSO at various concentrations were dispensed into a 384-well black OptiPlate using a Labcyte E...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent