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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
10
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Target
Potassium channel subfamily K member 3
(Homo sapiens (Human))
University Of Kansas Specialized Chemistry Center
Curated by
ChEMBL
Ligand
BDBM50123519
(2'-{[2-(4-Methoxy-phenyl)-acetylamino]-methyl}-bip...)
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Affinity Data
IC50: 7nM
Assay Description:
Inhibition of TASK-1 (unknown origin) expressed in CHO cells by thallium flux assay
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Target
Potassium channel subfamily K member 3
(Homo sapiens (Human))
University Of Kansas Specialized Chemistry Center
Curated by
ChEMBL
Ligand
BDBM50123519
(2'-{[2-(4-Methoxy-phenyl)-acetylamino]-methyl}-bip...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 7nM
Assay Description:
Inhibition of human TASK1 expressed in CHO cells by Inside-out macro-patches based electrophysiology assay
More data for this Ligand-Target Pair
Target Info
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Target
Potassium channel subfamily K member 3
(Homo sapiens (Human))
University Of Kansas Specialized Chemistry Center
Curated by
ChEMBL
Ligand
BDBM50123519
(2'-{[2-(4-Methoxy-phenyl)-acetylamino]-methyl}-bip...)
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Copy InChI
Affinity Data
IC50: 35nM
Assay Description:
Inhibition of human TASK-1 expressed in Xenopus laevis oocytes assessed as inhibition of channel current at +40mV holding potential by two-electrode ...
More data for this Ligand-Target Pair
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Target
Potassium channel subfamily K member 3
(Homo sapiens (Human))
University Of Kansas Specialized Chemistry Center
Curated by
ChEMBL
Ligand
BDBM50123519
(2'-{[2-(4-Methoxy-phenyl)-acetylamino]-methyl}-bip...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 35nM
Assay Description:
Inhibition of human TASK1 expressed in Xenopus oocytes by whole cell voltage clamp assay
More data for this Ligand-Target Pair
Target Info
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Target
Potassium channel subfamily K member 9
(Rattus norvegicus)
Universidad De Talca
Curated by
ChEMBL
Ligand
BDBM50123519
(2'-{[2-(4-Methoxy-phenyl)-acetylamino]-methyl}-bip...)
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Affinity Data
IC50: 36nM
Assay Description:
Inhibition of rat TASK3 expressed in (FRT) epithelial cells by chamber based electrophysiology assay
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Target
Potassium channel subfamily K member 9
(Homo sapiens (Human))
Universidad De Talca
Curated by
ChEMBL
Ligand
BDBM50123519
(2'-{[2-(4-Methoxy-phenyl)-acetylamino]-methyl}-bip...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 70nM
Assay Description:
Inhibition of human TASK3 expressed in CHO cells by Inside-out macro-patches based electrophysiology assay
More data for this Ligand-Target Pair
Target Info
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KEGG
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Target
Potassium channel subfamily K member 9
(Homo sapiens (Human))
Universidad De Talca
Curated by
ChEMBL
Ligand
BDBM50123519
(2'-{[2-(4-Methoxy-phenyl)-acetylamino]-methyl}-bip...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 318nM
Assay Description:
Inhibition of human TASK3 expressed in Xenopus oocytes by whole cell voltage clamp assay
More data for this Ligand-Target Pair
Target Info
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Target
Potassium voltage-gated channel subfamily A member 5
(Homo sapiens (Human))
Aventis Pharma Deutschland
Curated by
ChEMBL
Ligand
BDBM50123519
(2'-{[2-(4-Methoxy-phenyl)-acetylamino]-methyl}-bip...)
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Affinity Data
IC50: 1.20E+3nM
Assay Description:
Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytes
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Target
Potassium channel subfamily K member 17
(Homo sapiens)
Universidad De Talca
Curated by
ChEMBL
Ligand
BDBM50123519
(2'-{[2-(4-Methoxy-phenyl)-acetylamino]-methyl}-bip...)
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Affinity Data
IC50: 8.10E+3nM
Assay Description:
Inhibition of human TASK4 expressed in CHO cells by Inside-out macro-patches based electrophysiology assay
More data for this Ligand-Target Pair
Target Info
MMDB
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B.MOAD
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Target
Potassium channel subfamily K member 5
(Homo sapiens)
Universidad De Talca
Curated by
ChEMBL
Ligand
BDBM50123519
(2'-{[2-(4-Methoxy-phenyl)-acetylamino]-methyl}-bip...)
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Copy InChI
Affinity Data
IC50: 1.20E+4nM
Assay Description:
Inhibition of human TASK2 expressed in CHO cells by Inside-out macro-patches based electrophysiology assay
More data for this Ligand-Target Pair
Target Info
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CHEMBL
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