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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
30
hits in this display
Target
Proteasome subunit beta type-8
(Homo sapiens (Human))
Hangzhou Xixi Hospital
Curated by
ChEMBL
Ligand
BDBM50526811
(Kzr-616)
Copy SMILES
Copy InChI
Affinity Data
IC50: 0.0390nM
Assay Description:
Inhibition of 20S proteasome beta 5i (unknown origin) after 1 hr by fluorescence based assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
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In Depth
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Article
PubMed
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Target
Proteasome subunit beta type-10
(Homo sapiens (Human))
Hangzhou Xixi Hospital
Curated by
ChEMBL
Ligand
BDBM50526811
(Kzr-616)
Copy SMILES
Copy InChI
Affinity Data
IC50: 0.131nM
Assay Description:
Inhibition of 20S proteasome beta 2i (unknown origin) after 1 hr by fluorescence based assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
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In Depth
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PubMed
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Target
Proteasome subunit beta type-9
(Homo sapiens (Human))
Hangzhou Xixi Hospital
Curated by
ChEMBL
Ligand
BDBM50526811
(Kzr-616)
Copy SMILES
Copy InChI
Affinity Data
IC50: 0.623nM
Assay Description:
Inhibition of 20S proteasome beta 1i (unknown origin) after 1 hr by fluorescence based assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
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PC cid
PC sid
In Depth
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PubMed
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Target
Proteasome subunit beta type-5
(Homo sapiens (Human))
Hangzhou Xixi Hospital
Curated by
ChEMBL
Ligand
BDBM50526811
(Kzr-616)
Copy SMILES
Copy InChI
Affinity Data
IC50: 0.688nM
Assay Description:
Inhibition of 20S proteasome beta 5c (unknown origin) after 1 hr by fluorescence based assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
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PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-2
(Homo sapiens (Human))
Hangzhou Xixi Hospital
Curated by
ChEMBL
Ligand
BDBM50526811
(Kzr-616)
Copy SMILES
Copy InChI
Affinity Data
IC50: 28nM
Assay Description:
Inhibition of 20S proteasome beta 2c (unknown origin) after 1 hr by fluorescence based assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-8
(Homo sapiens (Human))
Hangzhou Xixi Hospital
Curated by
ChEMBL
Ligand
BDBM50526811
(Kzr-616)
Copy SMILES
Copy InChI
Affinity Data
IC50: 39nM
Assay Description:
Inhibition of LMP7 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-8
(Homo sapiens (Human))
Hangzhou Xixi Hospital
Curated by
ChEMBL
Ligand
BDBM50526811
(Kzr-616)
Copy SMILES
Copy InChI
Affinity Data
IC50: 39nM
Assay Description:
Inhibition of LMP7 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-8
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526811
(Kzr-616)
Copy SMILES
Copy InChI
Affinity Data
IC50: 57nM
Assay Description:
Inhibition of LMP7 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-8
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526811
(Kzr-616)
Copy SMILES
Copy InChI
Affinity Data
IC50: 57nM
Assay Description:
Inhibition of LMP7 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-9
(Homo sapiens (Human))
Hangzhou Xixi Hospital
Curated by
ChEMBL
Ligand
BDBM50526811
(Kzr-616)
Copy SMILES
Copy InChI
Affinity Data
IC50: 131nM
Assay Description:
Inhibition of LMP2 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-9
(Homo sapiens (Human))
Hangzhou Xixi Hospital
Curated by
ChEMBL
Ligand
BDBM50526811
(Kzr-616)
Copy SMILES
Copy InChI
Affinity Data
IC50: 131nM
Assay Description:
Inhibition of LMP2 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-9
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526811
(Kzr-616)
Copy SMILES
Copy InChI
Affinity Data
IC50: 179nM
Assay Description:
Inhibition of LMP2 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-9
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526811
(Kzr-616)
Copy SMILES
Copy InChI
Affinity Data
IC50: 179nM
Assay Description:
Inhibition of LMP2 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-1
(Homo sapiens (Human))
Hangzhou Xixi Hospital
Curated by
ChEMBL
Ligand
BDBM50526811
(Kzr-616)
Copy SMILES
Copy InChI
Affinity Data
IC50: 430nM
Assay Description:
Inhibition of 20S proteasome beta 1c (unknown origin) after 1 hr by fluorescence based assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-5
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526811
(Kzr-616)
Copy SMILES
Copy InChI
Affinity Data
IC50: 483nM
Assay Description:
Inhibition of 20S proteosome beta 5 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-5
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526811
(Kzr-616)
Copy SMILES
Copy InChI
Affinity Data
IC50: 483nM
Assay Description:
Inhibition of 20S proteosome beta 5 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-10
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526811
(Kzr-616)
Copy SMILES
Copy InChI
Affinity Data
IC50: 522nM
Assay Description:
Inhibition of MECL1 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-10
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526811
(Kzr-616)
Copy SMILES
Copy InChI
Affinity Data
IC50: 522nM
Assay Description:
Inhibition of MECL1 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-2
(Homo sapiens (Human))
Hangzhou Xixi Hospital
Curated by
ChEMBL
Ligand
BDBM50526811
(Kzr-616)
Copy SMILES
Copy InChI
Affinity Data
IC50: 604nM
Assay Description:
Inhibition of 20S proteosome beta 2 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-2
(Homo sapiens (Human))
Hangzhou Xixi Hospital
Curated by
ChEMBL
Ligand
BDBM50526811
(Kzr-616)
Copy SMILES
Copy InChI
Affinity Data
IC50: 604nM
Assay Description:
Inhibition of 20S proteosome beta 2 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-10
(Homo sapiens (Human))
Hangzhou Xixi Hospital
Curated by
ChEMBL
Ligand
BDBM50526811
(Kzr-616)
Copy SMILES
Copy InChI
Affinity Data
IC50: 623nM
Assay Description:
Inhibition of MECL1 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-10
(Homo sapiens (Human))
Hangzhou Xixi Hospital
Curated by
ChEMBL
Ligand
BDBM50526811
(Kzr-616)
Copy SMILES
Copy InChI
Affinity Data
IC50: 623nM
Assay Description:
Inhibition of MECL1 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-5
(Homo sapiens (Human))
Hangzhou Xixi Hospital
Curated by
ChEMBL
Ligand
BDBM50526811
(Kzr-616)
Copy SMILES
Copy InChI
Affinity Data
IC50: 688nM
Assay Description:
Inhibition of 20S proteosome beta 5 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-5
(Homo sapiens (Human))
Hangzhou Xixi Hospital
Curated by
ChEMBL
Ligand
BDBM50526811
(Kzr-616)
Copy SMILES
Copy InChI
Affinity Data
IC50: 688nM
Assay Description:
Inhibition of 20S proteosome beta 5 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-2
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526811
(Kzr-616)
Copy SMILES
Copy InChI
Affinity Data
IC50: 857nM
Assay Description:
Inhibition of 20S proteosome beta 2 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-2
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526811
(Kzr-616)
Copy SMILES
Copy InChI
Affinity Data
IC50: 857nM
Assay Description:
Inhibition of 20S proteosome beta 2 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-1
(Homo sapiens (Human))
Hangzhou Xixi Hospital
Curated by
ChEMBL
Ligand
BDBM50526811
(Kzr-616)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.06E+4nM
Assay Description:
Inhibition of 20S proteosome beta 1 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-1
(Homo sapiens (Human))
Hangzhou Xixi Hospital
Curated by
ChEMBL
Ligand
BDBM50526811
(Kzr-616)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.06E+4nM
Assay Description:
Inhibition of 20S proteosome beta 1 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-1
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526811
(Kzr-616)
Copy SMILES
Copy InChI
Affinity Data
IC50: >2.50E+4nM
Assay Description:
Inhibition of 20S proteosome beta 1 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-1
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526811
(Kzr-616)
Copy SMILES
Copy InChI
Affinity Data
IC50: >2.50E+4nM
Assay Description:
Inhibition of 20S proteosome beta 1 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI