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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Prostaglandin D2 receptor 2
(Homo sapiens (Human))
7Tm Pharma
Curated by
ChEMBL
Ligand
BDBM50200247
(4-bromo-2-[1-(4-methoxyphenyl)-1H-pyrazole-4-carbo...)
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Affinity Data
IC50: 3.60nM
Assay Description:
Displacement of [3H]PGD2 from human CRTH2 receptor expressed in HEK293 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
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In Depth
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Article
PubMed
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Target
Prostaglandin D2 receptor 2
(Homo sapiens (Human))
7Tm Pharma
Curated by
ChEMBL
Ligand
BDBM50200247
(4-bromo-2-[1-(4-methoxyphenyl)-1H-pyrazole-4-carbo...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 53nM
Assay Description:
Antagonist activity against CRTH2 receptor measured as inhibition of PGD2-induced beta-arrestin translocation in HEK293 cells by BRET assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI