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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
13
hits in this display
Target
Poly [ADP-ribose] polymerase tankyrase-1/tankyrase-2
(Homo sapiens (Human))
University Of Oulu
Curated by
ChEMBL
Ligand
BDBM50136755
(CHEMBL3752386)
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Affinity Data
IC50: 360nM
Assay Description:
Inhibition of tankyrase in WNT3a-stimulated human HEK293 cells by luciferase reporter gene assay
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
PubMed
PDB
3D Structure (crystal)
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Target
Poly [ADP-ribose] polymerase tankyrase-1
(Homo sapiens (Human))
University Of Oulu
Curated by
ChEMBL
Ligand
BDBM50136755
(CHEMBL3752386)
Copy SMILES
Copy InChI
Affinity Data
IC50: 562nM
Assay Description:
Inhibition of human TNKS1 by fluorescence analysis
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
PubMed
PDB
3D Structure (crystal)
Copy BDB DOI
Target
Poly [ADP-ribose] polymerase tankyrase-1
(Homo sapiens (Human))
University Of Oulu
Curated by
ChEMBL
Ligand
BDBM50136755
(CHEMBL3752386)
Copy SMILES
Copy InChI
Affinity Data
IC50: 570nM
Assay Description:
Inhibition of human TNKS1 by fluorescence analysis
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
PubMed
PDB
3D Structure (crystal)
Copy BDB DOI
Target
Poly [ADP-ribose] polymerase tankyrase-2
(Homo sapiens (Human))
University Of Oulu
Curated by
ChEMBL
Ligand
BDBM50136755
(CHEMBL3752386)
Copy SMILES
Copy InChI
Affinity Data
IC50: 2.14E+3nM
Assay Description:
Inhibition of human TNKS2 by fluorescence analysis
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
PubMed
PDB
3D Structure (crystal)
Copy BDB DOI
Target
Poly [ADP-ribose] polymerase tankyrase-2
(Homo sapiens (Human))
University Of Oulu
Curated by
ChEMBL
Ligand
BDBM50136755
(CHEMBL3752386)
Copy SMILES
Copy InChI
Affinity Data
IC50: 2.15E+3nM
Assay Description:
Inhibition of human TNKS2 by fluorescence analysis
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
PubMed
PDB
3D Structure (crystal)
Copy BDB DOI
Target
Protein mono-ADP-ribosyltransferase PARP14
(Homo sapiens (Human))
University Of Oulu
Curated by
ChEMBL
Ligand
BDBM50136755
(CHEMBL3752386)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of human ARTD8 by fluorescence analysis
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
PubMed
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Target
Protein mono-ADP-ribosyltransferase PARP12
(Homo sapiens (Human))
University Of Oulu
Curated by
ChEMBL
Ligand
BDBM50136755
(CHEMBL3752386)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of human ARTD12 by fluorescence analysis
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
PubMed
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Target
Protein mono-ADP-ribosyltransferase PARP10
(Homo sapiens (Human))
University Of Oulu
Curated by
ChEMBL
Ligand
BDBM50136755
(CHEMBL3752386)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of human ARTD10 by fluorescence analysis
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
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CHEMBL
PC cid
PC sid
PDB
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In Depth
Details
Article
PubMed
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Target
Protein mono-ADP-ribosyltransferase PARP15
(Homo sapiens (Human))
University Of Oulu
Curated by
ChEMBL
Ligand
BDBM50136755
(CHEMBL3752386)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of human ARTD7 by fluorescence analysis
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
PubMed
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Target
Protein mono-ADP-ribosyltransferase PARP4
(Homo sapiens (Human))
University Of Oulu
Curated by
ChEMBL
Ligand
BDBM50136755
(CHEMBL3752386)
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Affinity Data
IC50: >1.00E+5nM
Assay Description:
Inhibition of human ARTD4 by fluorescence analysis
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
PubMed
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Target
Protein mono-ADP-ribosyltransferase PARP3 [R100H]
(Homo sapiens (Human))
University Of Oulu
Curated by
ChEMBL
Ligand
BDBM50136755
(CHEMBL3752386)
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Affinity Data
IC50: >1.00E+5nM
Assay Description:
Inhibition of human ARTD3 by fluorescence analysis
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
PubMed
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Target
Poly [ADP-ribose] polymerase 1
(Homo sapiens (Human))
University Of Oulu
Curated by
ChEMBL
Ligand
BDBM50136755
(CHEMBL3752386)
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Copy InChI
Affinity Data
IC50: >1.00E+5nM
Assay Description:
Inhibition of human ARTD1 by fluorescence analysis
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Poly [ADP-ribose] polymerase 2
(Homo sapiens (Human))
University Of Oulu
Curated by
ChEMBL
Ligand
BDBM50136755
(CHEMBL3752386)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+5nM
Assay Description:
Inhibition of human ARTD2 by fluorescence analysis
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI