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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Endoplasmic reticulum aminopeptidase 1
(Homo sapiens (Human))
Kansas University Specialized Chemistry Center
Curated by
ChEMBL
Ligand
BDBM50519953
(CHEMBL2140832)
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Affinity Data
Ki: 3.80E+3nM
Assay Description:
Competitive inhibition of recombinant human C-terminal His6-tagged ERAP1 expressed in baculovirus infected BTA-TN-5B1-4 insect cells using varying le...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
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In Depth
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Article
PubMed
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Target
Endoplasmic reticulum aminopeptidase 1
(Homo sapiens (Human))
Kansas University Specialized Chemistry Center
Curated by
ChEMBL
Ligand
BDBM50519953
(CHEMBL2140832)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.00E+3nM
Assay Description:
Inhibition of ERAP1 in human HeLa cells stably expressing H-2 Kb infected with vaccinia virus containing ss-LEQLE-SIINFEKL epitope assessed as suppre...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Endoplasmic reticulum aminopeptidase 1
(Homo sapiens (Human))
Kansas University Specialized Chemistry Center
Curated by
ChEMBL
Ligand
BDBM50519953
(CHEMBL2140832)
Copy SMILES
Copy InChI
Affinity Data
IC50: 5.30E+3nM
Assay Description:
Inhibition of recombinant human C-terminal His6-tagged ERAP1 expressed in baculovirus infected BTA-TN-5B1-4 insect cells using WRCYEKMALK as substrat...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Endoplasmic reticulum aminopeptidase 2
(Homo sapiens (Human))
Kansas University Specialized Chemistry Center
Curated by
ChEMBL
Ligand
BDBM50519953
(CHEMBL2140832)
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Copy InChI
Affinity Data
IC50: >2.00E+5nM
Assay Description:
Inhibition of recombinant human C-terminal His6-tagged ERAP2 expressed in baculovirus infected BTA-TN-5B1-4 insect cells using R-AMC as substrate mea...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI