Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL

LigandBDBM50375434(CHEMBL407371)Copy SMILESCopy InChI

Affinity DataIC50:  0.980nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL

LigandBDBM50375434(CHEMBL407371)Copy SMILESCopy InChI

Affinity DataEC50:  0.740nMAssay Description:Agonist activity at human PRB expressed in CHO cellsMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI