Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50497605(CHEMBL3356163)
Affinity DataIC50:  40nMAssay Description:Inhibition of integrin alphavbeta3 (unknown origin)-mediated K562 cell adhesion to LAPb1 coated surface by fluorescence analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50497605(CHEMBL3356163)
Affinity DataIC50:  63nMAssay Description:Inhibition of integrin alphavbeta5 (unknown origin)-mediated K562 cell adhesion to vitronectin coated surface by fluorescence analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-6(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50497605(CHEMBL3356163)
Affinity DataIC50:  316nMAssay Description:Inhibition of integrin alphavbeta6 (unknown origin)-mediated K562 cell adhesion to LAPb1 coated surface by fluorescence analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-8(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50497605(CHEMBL3356163)
Affinity DataIC50:  501nMAssay Description:Inhibition of integrin alphavbeta8 (unknown origin)-mediated K562 cell adhesion to LAPb1 coated surface by fluorescence analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed