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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Prostaglandin D2 receptor 2
(Homo sapiens (Human))
RhôNe-Poulenc Rorer
Curated by
ChEMBL
Ligand
BDBM50444781
(CHEMBL3099118)
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Affinity Data
IC50: 4nM
Assay Description:
Antagonist activity at CRTh2 in human RBC assessed as inhibition of PGD2-induced eosinophil shape change
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Prostaglandin D2 receptor 2
(Homo sapiens (Human))
RhôNe-Poulenc Rorer
Curated by
ChEMBL
Ligand
BDBM50444781
(CHEMBL3099118)
Copy SMILES
Copy InChI
Affinity Data
IC50: 30nM
Assay Description:
Antagonist activity at CRTh2 (unknown origin) expressed in CHO.K1 cells assessed as inhibition of PGD2-induced [35S]-GTPgammaS binding after 2 hrs by...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Prostaglandin D2 receptor 2
(Homo sapiens (Human))
RhôNe-Poulenc Rorer
Curated by
ChEMBL
Ligand
BDBM50444781
(CHEMBL3099118)
Copy SMILES
Copy InChI
Affinity Data
IC50: 50nM
Assay Description:
Antagonist activity at CRTh2 in human whole blood assessed as inhibition of PGD2-induced eosinophil shape change
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Prostaglandin D2 receptor 2
(Homo sapiens (Human))
RhôNe-Poulenc Rorer
Curated by
ChEMBL
Ligand
BDBM50444781
(CHEMBL3099118)
Copy SMILES
Copy InChI
Affinity Data
IC50: 70nM
Assay Description:
Antagonist activity at CRTh2 (unknown origin) expressed in CHO.K1 cells assessed as inhibition of PGD2-induced [35S]-GTPgammaS binding after 2 hrs by...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI