Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 12 hits in this display
BDBM270506(3-[({(1S)-5-[2-methyl-4-(2,2,2-trifluoroethoxy)phe...)
BDBM270506(3-[({(1S)-5-[2-methyl-4-(2,2,2-trifluoroethoxy)phe...)
IC50: <100nMAssay Description:Jarid1b: The ability of test compounds to inhibit the activity of Jarid1B was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
BDBM270506(3-[({(1S)-5-[2-methyl-4-(2,2,2-trifluoroethoxy)phe...)
BDBM270506(3-[({(1S)-5-[2-methyl-4-(2,2,2-trifluoroethoxy)phe...)
BDBM270506(3-[({(1S)-5-[2-methyl-4-(2,2,2-trifluoroethoxy)phe...)
BDBM270506(3-[({(1S)-5-[2-methyl-4-(2,2,2-trifluoroethoxy)phe...)
BDBM270506(3-[({(1S)-5-[2-methyl-4-(2,2,2-trifluoroethoxy)phe...)
BDBM270506(3-[({(1S)-5-[2-methyl-4-(2,2,2-trifluoroethoxy)phe...)
BDBM270506(3-[({(1S)-5-[2-methyl-4-(2,2,2-trifluoroethoxy)phe...)
IC50: 5.50E+3nMAssay Description:JMJD3: The enzymatic assay of JMJD3 activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of t...More data for this Ligand-Target Pair
BDBM270506(3-[({(1S)-5-[2-methyl-4-(2,2,2-trifluoroethoxy)phe...)
IC50: 5.50E+3nMAssay Description:JMJD2C: The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditio...More data for this Ligand-Target Pair
BDBM270506(3-[({(1S)-5-[2-methyl-4-(2,2,2-trifluoroethoxy)phe...)
BDBM270506(3-[({(1S)-5-[2-methyl-4-(2,2,2-trifluoroethoxy)phe...)