Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetProtein-arginine deiminase type-3(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50535201(CHEMBL4442207)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of recombinant human 6His-tagged PAD3 expressed in Escherichia coli BL21-DE3 pLysS assessed as reduction in residual activity preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-4(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50535201(CHEMBL4442207)
Affinity DataIC50:  3.60E+4nMAssay Description:Inhibition of recombinant human GST-tagged PAD4 expressed in Escherichia coli BL21-DE3 pLysS assessed as reduction in reduction in residual activity ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-2(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50535201(CHEMBL4442207)
Affinity DataIC50:  1.51E+5nMAssay Description:Inhibition of recombinant human 6His-tagged PAD2 assessed as reduction in residual activity preincubated for 15 mins followed by addition of N-benzoy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-1(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50535201(CHEMBL4442207)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of recombinant human 6His-tagged PAD1 assessed as reduction in residual activity preincubated for 15 mins followed by addition of N-benzoy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed