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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 7 hits in this display   

TargetCoagulation factor X(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50386271(CHEMBL2040983)
Affinity DataIC50:  270nMAssay Description:Inhibition of human factor 10a using chromogenic spectrozyme F10a as substrate after 10 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50386271(CHEMBL2040983)
Affinity DataIC50:  7.53E+4nMAssay Description:Inhibition of bovine alpha-chymotrypsin using chromogenic spectrozyme CTY as substrate after 10 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50386271(CHEMBL2040983)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of human factor 2a using chromogenic spectrozyme TH as substrate after 10 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50386271(CHEMBL2040983)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of human factor 11a using chromogenic S2366 as substrate after 10 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XII(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50386271(CHEMBL2040983)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of factor 12a using chromogenic spectrozyme 12a as substrate after 10 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50386271(CHEMBL2040983)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of human factor 7a using chromogenic spectrozyme 7a as substrate after 10 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor IX(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50386271(CHEMBL2040983)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of human factor 9a using chromogenic spectrozyme 9a as substrate after 10 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed