Home
About
Info
Download
WebServices
Contact
Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Potassium channel subfamily K member 3
(Homo sapiens (Human))
Sanofi
US Patent
Ligand
BDBM218364
(US9284333, 16dh | US9884860, Example 16dh)
Copy SMILES
Copy InChI
Affinity Data
IC50: 290nM
T: 2°C
Assay Description:
Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Potassium channel subfamily K member 3
(Homo sapiens (Human))
Sanofi
US Patent
Ligand
BDBM218364
(US9284333, 16dh | US9884860, Example 16dh)
Copy SMILES
Copy InChI
Affinity Data
IC50: 290nM
T: 2°C
Assay Description:
Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliculated. Subsequently,...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Potassium voltage-gated channel subfamily H member 2
(Homo sapiens (Human))
Sanofi
US Patent
Ligand
BDBM218364
(US9284333, 16dh | US9884860, Example 16dh)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
T: 2°C
Assay Description:
The effect of compounds of the formula I on the cloned human cardiac hERG channel was evaluated in an in vitro model using a whole-cell patch-clampin...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI