Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 12 hits in this display
IC50: 13nMAssay Description:Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR...More data for this Ligand-Target Pair
Kd: 1.50E+3nMAssay Description:Binding affinity to CK1 in Plasmodium falciparum 3D7 blood stage extract incubated for 1 hr by kinobeads based pull down assayMore data for this Ligand-Target Pair
Kd: 60nMAssay Description:Binding affinity to CDPK4 in Plasmodium falciparum 3D7 blood stage extract incubated for 1 hr by kinobeads based pull down assayMore data for this Ligand-Target Pair
Kd: 2.10E+3nMAssay Description:Binding affinity to CDPK1 in Plasmodium falciparum 3D7 blood stage extract incubated for 1 hr in presence of ATP-competitive kinase inhibitor by kino...More data for this Ligand-Target Pair
Kd: 2.10E+3nMAssay Description:Binding affinity to CDPK1 in Plasmodium falciparum 3D7 blood stage extract incubated for 1 hr by kinobeads based pull down assayMore data for this Ligand-Target Pair
Kd: 60nMAssay Description:Binding affinity to CDPK4 in Plasmodium falciparum 3D7 blood stage extract incubated for 1 hr by kinobeads based pull down assayMore data for this Ligand-Target Pair
Kd: 2.10E+3nMAssay Description:Binding affinity to CDPK1 in Plasmodium falciparum 3D7 blood stage extract incubated for 1 hr by kinobeads based pull down assayMore data for this Ligand-Target Pair
Kd: 1.50E+3nMAssay Description:Binding affinity to CK1 in Plasmodium falciparum 3D7 blood stage extract incubated for 1 hr by kinobeads based pull down assayMore data for this Ligand-Target Pair
Kd: 60nMAssay Description:Binding affinity to CDPK4 in Plasmodium falciparum 3D7 blood stage extract incubated for 1 hr in presence of ATP-competitive kinase inhibitor by kino...More data for this Ligand-Target Pair