Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetProteasome subunit beta type-8(Homo sapiens (Human))
Weill Cornell Medicine

Curated by ChEMBL
LigandPNGBDBM50587109(CHEMBL5079787)
Affinity DataIC50:  69nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunit using Suc-LLVY-AMC as substrate measured over 1.5 to 2 hrs by plate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Weill Cornell Medicine

Curated by ChEMBL
LigandPNGBDBM50587109(CHEMBL5079787)
Affinity DataIC50:  73nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5c subunit using Suc-LLVY-AMC as substrate measured over 1.5 to 2 hrs by plate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-10(Homo sapiens (Human))
Weill Cornell Medicine

Curated by ChEMBL
LigandPNGBDBM50587109(CHEMBL5079787)
Affinity DataIC50:  4.45E+4nMAssay Description:Inhibition of human 20S immunoproteasome beta-2i subunit using Z-VLR-AMC as substrate measured over 1.5 to 2 hrs by plate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed