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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetCarboxypeptidase B(Homo sapiens (Human))
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296421(2-(4-benzyl-5-(thiophen-2-yl)-4H-1,2,4-triazol-3-y...)
Affinity DataKi:  1.16E+4nMAssay Description:Inhibition of human recombinant carboxypeptidase B expressed in Pichia pastoris systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B(Helicoverpa zea (Corn earworm moth) (Heliothis zea...)
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296421(2-(4-benzyl-5-(thiophen-2-yl)-4H-1,2,4-triazol-3-y...)
Affinity DataKi:  2.72E+4nMAssay Description:Inhibition of corn earworm recombinant carboxypeptidase B expressed in Pichia pastoris systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase A1(Bos taurus (bovine))
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296421(2-(4-benzyl-5-(thiophen-2-yl)-4H-1,2,4-triazol-3-y...)
Affinity DataKi:  1.55E+5nMAssay Description:Inhibition of bovine carboxypeptidase A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed