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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Calmodulin-domain protein kinase 1
(Toxoplasma gondii)
University of Washington Through Its Center For Commercialization
US Patent
Ligand
BDBM286281
(US9518026, Example 74 | US9956214, Compound 1657)
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Affinity Data
IC50: 3nM
Assay Description:
Inhibition of TgCDPK1 and CpCDPK1 was determined using a luminescent kinase assay which measures ATP depletion in the presence of the Syntide 2 pepti...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/TrEMBL
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Uncharacterized protein
(Cryptosporidium parvum)
University of Washington Through Its Center For Commercialization
US Patent
Ligand
BDBM286281
(US9518026, Example 74 | US9956214, Compound 1657)
Copy SMILES
Copy InChI
Affinity Data
IC50: 4nM
Assay Description:
Inhibition of TgCDPK1 and CpCDPK1 was determined using a luminescent kinase assay which measures ATP depletion in the presence of the Syntide 2 pepti...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/TrEMBL
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Calcium-dependent protein kinase 1
(Cryptosporidium parvum)
University of Washington Through Its Center For Commercialization
US Patent
Ligand
BDBM286281
(US9518026, Example 74 | US9956214, Compound 1657)
Copy SMILES
Copy InChI
Affinity Data
IC50: 5nM
Assay Description:
Inhibition of TgCDPK1 and CpCDPK1 was determined using a luminescent kinase assay which measures ATP depletion in the presence of the Syntide 2 pepti...
More data for this Ligand-Target Pair
Target Info
UniProtKB/TrEMBL
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Calmodulin-domain protein kinase 1
(Toxoplasma gondii)
University of Washington Through Its Center For Commercialization
US Patent
Ligand
BDBM286281
(US9518026, Example 74 | US9956214, Compound 1657)
Copy SMILES
Copy InChI
Affinity Data
IC50: 12nM
Assay Description:
Inhibition of TgCDPK1 and CpCDPK1 was determined using a luminescent kinase assay which measures ATP depletion in the presence of the Syntide 2 pepti...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/TrEMBL
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Found 4 hits in this display