Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 8 hits in this display
BDBM141087(US11547697, Compound 487 | US9682141, 487)
BDBM141087(US11547697, Compound 487 | US9682141, 487)
IC50: >1.00E+4nMT: 2°CAssay Description:Briefly, the assay is a time resolved FRET assay that indirectly measures PIP3 product formed by the activity of a PI3-K. The kinase reaction is perf...More data for this Ligand-Target Pair
BDBM141087(US11547697, Compound 487 | US9682141, 487)
IC50: >1.00E+4nMT: 2°CAssay Description:Briefly, the assay is a time resolved FRET assay that indirectly measures PIP3 product formed by the activity of a PI3-K. The kinase reaction is perf...More data for this Ligand-Target Pair
BDBM141087(US11547697, Compound 487 | US9682141, 487)
BDBM141087(US11547697, Compound 487 | US9682141, 487)
IC50: >1.00E+4nMAssay Description:An exemplary system is PI 3-Kinase (human) HTRF? Assay from Upstate. The assay can be carried out according to the procedures suggested by the manufa...More data for this Ligand-Target Pair
BDBM141087(US11547697, Compound 487 | US9682141, 487)
IC50: >1.00E+4nMAssay Description:An exemplary system is PI 3-Kinase (human) HTRF? Assay from Upstate. The assay can be carried out according to the procedures suggested by the manufa...More data for this Ligand-Target Pair
BDBM141087(US11547697, Compound 487 | US9682141, 487)
IC50: >1.00E+4nMAssay Description:An exemplary system is PI 3-Kinase (human) HTRF? Assay from Upstate. The assay can be carried out according to the procedures suggested by the manufa...More data for this Ligand-Target Pair
BDBM141087(US11547697, Compound 487 | US9682141, 487)
IC50: >1.00E+4nMT: 2°CAssay Description:Briefly, the assay is a time resolved FRET assay that indirectly measures PIP3 product formed by the activity of a PI3-K. The kinase reaction is perf...More data for this Ligand-Target Pair