Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))TBA
LigandPNGBDBM50460478(CHEMBL4226903)
Affinity DataIC50:  7.40E+4nMAssay Description:Antagonist activity at adrenergic Alpha-1B receptor in guinea pig spleenMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))TBA
LigandPNGBDBM50460478(CHEMBL4226903)
Affinity DataIC50:  8.90E+4nMAssay Description:Antagonist activity at adrenergic Alpha-1B receptor in guinea pig spleenMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed
TargetADP-ribose glycohydrolase MACROD2(Homo sapiens)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50460478(CHEMBL4226903)
Affinity DataKd:  150nMAssay Description:Binding affinity to human MDO2 by ITCMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetADP-ribose glycohydrolase MACROD1(Homo sapiens)
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50460478(CHEMBL4226903)
Affinity DataKd:  900nMAssay Description:Binding affinity to human MDO1 by ITCMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed