Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetProgesterone receptor(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50359653(CHEMBL1928869)
Affinity DataIC50:  1.60E+3nMAssay Description:Displacement of [3H]progestrone from PRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMineralocorticoid receptor(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50359653(CHEMBL1928869)
Affinity DataIC50:  2.00E+3nMAssay Description:Displacement of [3H]aldosterone from cytosolic human MR expressed in HEK293 cells after 16 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50359653(CHEMBL1928869)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]dexomethasone from GRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50359653(CHEMBL1928869)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]testosterone from ARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed