Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50385620(CHEMBL2042238)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]PGD2 from human CRTH2 receptor expressed in CHO cells after 90 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50385620(CHEMBL2042238)
Affinity DataIC50:  7.40nMAssay Description:Antagonist activity at CRTH2 receptor in human whole blood assessed as inhibition of PGD2-induced eosinophil chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50385620(CHEMBL2042238)
Affinity DataIC50:  69nMAssay Description:Antagonist activity at CRTH2 receptor in human whole blood assessed as inhibition of PGD2-induced eosinophil shape change pretreated for 20 mins meas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed