Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50200258(2-(1-phenyl-1H-pyrazole-4-carbonyl)phenoxyacetic a...)
Affinity DataIC50:  510nMAssay Description:Displacement of [3H]PGD2 from human CRTH2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50200258(2-(1-phenyl-1H-pyrazole-4-carbonyl)phenoxyacetic a...)
Affinity DataIC50:  5.35E+3nMAssay Description:Antagonist activity against CRTH2 receptor measured as inhibition of PGD2-induced beta-arrestin translocation in HEK293 cells by BRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed