Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50309273(2-(2-benzhydryl-4-(4-chlorophenyl)thiazol-5-yl)ace...)
Affinity DataIC50:  14nMAssay Description:Displacement of[3H]PGD2 from human CRTH2 receptor expressed in HEK385-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50309273(2-(2-benzhydryl-4-(4-chlorophenyl)thiazol-5-yl)ace...)
Affinity DataIC50:  60nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in HEK285-7 cells assessed as inhibition of beta arrestin translocation by bioluminescence reso...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor(Homo sapiens (Human))
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50309273(2-(2-benzhydryl-4-(4-chlorophenyl)thiazol-5-yl)ace...)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of DP1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed